SCHEMBL2943307

SCHEMBL2943307

CCNNC(=O)NCCc1ccc(-c2ccccc2CC)cc1F

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.45
FFAR4 Q5NUL3 1/20 0.45
HIF1A Q16665 3/20 0.42
BDKRB1 P46663 10/20 0.42
ABL1 P00519 2/20 0.42
CNR1 P21554 1/20 0.40
ALOX5AP P20292 1/20 0.40
FEN1 P39748 1/20 0.40
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2943098 0.99 FFAR1 (0.45) FFAR1FFAR4HIF1ABDKRB1ABL1
SCHEMBL3655943 0.77 EPHX2 (0.46) CNR1KMT2A
SCHEMBL2949321 0.75 ALOX5AP (0.53) FFAR1FFAR4BDKRB1ALOX5APFEN1
SCHEMBL2950599 0.74 BDKRB1 (0.74) BDKRB1CNR1
SCHEMBL2948017 0.73 ALOX5AP (0.54) FFAR1FFAR4BDKRB1ALOX5APFEN1
SCHEMBL2943305 0.70 FFAR1 (0.45) FFAR1FFAR4BDKRB1ABL1ALOX5AP
SCHEMBL23347204 0.70 ALOX5AP (0.56) FFAR1FFAR4ALOX5APFEN1
SCHEMBL5925998 0.69 HIF1A (0.50) HIF1AKMT2A
SCHEMBL2942746 0.69 BDKRB1 (0.49) FFAR1FFAR4BDKRB1ALOX5APFEN1
Hydrochloric Acid SCHEMBL2943097 0.69 FFAR1 (0.44) FFAR1FFAR4BDKRB1ABL1ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396301-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS Jerini AG (DE) 2011-12-21 EP disclosed
WO-2010091876-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS JERINI AG (DE) 2010-08-19 WO disclosed