SCHEMBL2949321

SCHEMBL2949321

CCc1ccccc1-c1ccc(CCN)c(F)c1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 6/20 0.53
FEN1 P39748 6/20 0.53
TAAR1 Q96RJ0 3/20 0.50
FFAR1 O14842 1/20 0.47
FFAR4 Q5NUL3 1/20 0.47
ADRA2C P18825 1/20 0.46
TRPA1 O75762 1/20 0.43
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
LTB4R2 Q9NPC1 1/20 0.40
CSNK2A2 P19784 1/20 0.40
CSNK2B P67870 1/20 0.40
CSNK2A1 P68400 1/20 0.40
CSNK2A3 Q8NEV1 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
BDKRB1 P46663 1/20 0.40
HTR7 P34969 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2948017 0.89 ALOX5AP (0.54) ALOX5APFEN1FFAR1FFAR4TRPA1
SCHEMBL23347204 0.82 ALOX5AP (0.56) ALOX5APFEN1FFAR1FFAR4TRPA1
SCHEMBL15060621 0.78 ALOX5AP (0.46) ALOX5APFEN1TAAR1LTB4R2
SCHEMBL2943305 0.76 FFAR1 (0.45) ALOX5APFEN1FFAR1FFAR4LTB4R2
SCHEMBL9287992 0.76 ALOX5AP (0.50) ALOX5APFEN1FFAR1FFAR4TRPA1
SCHEMBL2949319 0.76 ALOX5AP (0.54) ALOX5APFEN1TRPA1PDE3BPDE3A
Hydrochloric Acid SCHEMBL2943097 0.76 FFAR1 (0.44) ALOX5APFEN1FFAR1FFAR4LTB4R2
SCHEMBL2950123 0.75 ALOX5AP (0.50) ALOX5APFEN1FFAR1FFAR4TRPA1
SCHEMBL2943307 0.75 FFAR1 (0.45) ALOX5APFEN1FFAR1FFAR4BDKRB1
SCHEMBL9289358 0.74 PTGS2 (0.57) ALOX5APFEN1TRPA1PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396301-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS Jerini AG (DE) 2011-12-21 EP disclosed
WO-2010091876-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS JERINI AG (DE) 2010-08-19 WO disclosed