Bgc-20-1531 Free Base

Bgc-20-1531 Free Base

SCHEMBL29433722

COc1ccc(-c2ccc(OCc3cc(C(=O)NS(=O)(=O)c4ccccc4C)oc3C)cc2)nc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 20/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bgc-20-1531 Free Base SCHEMBL2348089 1.00 PTGER4 (1.00) PTGER4
SCHEMBL3534655 0.90 PTGER4 (1.00) PTGER4
SCHEMBL3532327 0.89 PTGER4 (0.81) PTGER4
SCHEMBL3541275 0.86 PTGER4 (0.80) PTGER4
Bgc-20-1531 Free Base SCHEMBL29508262 0.84 PTGER4 (1.00) PTGER4
SCHEMBL4688621 0.84 PTGER4 (1.00) PTGER4
Bgc-20-1531 Free Base SCHEMBL30114901 0.84 PTGER4 (1.00) PTGER4
Bgc-20-1531 Free Base SCHEMBL2355810 0.84 PTGER4 (1.00) PTGER4
SCHEMBL4689376 0.83 PTGER4 (0.87) PTGER4
SCHEMBL14271689 0.81 PTGER4 (0.71) PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4656246-A2 COMBINATION THERAPIES FOR THE TREATMENT OF CANCER Eisai R&D Management Co., Ltd. (JP) 2025-12-03 EP disclosed
EP-3134085-B1 COMBINATION THERAPIES FOR THE TREATMENT OF CANCER EISAI R&D MAN CO LTD (JP) 2025-07-02 EP disclosed
US-12240860-B2 Heterobicyclic carboxylic acids and salts thereof Foshan Ionova Biotherapeutics Co., Inc. (CN) 2025-03-04 US disclosed
US-20240285640-A1 COMBINATION THERAPY FOR TREATING PIK3CA-MUTATED CANCER ADLAI NORTYE BIOPHARMA CO., LTD. (CN) 2024-08-29 US disclosed
CN-111936502-B Heterobicyclic carboxylic acids and salts thereof 深圳市原力生命科学有限公司 2024-05-31 CN disclosed
US-20230390303-A1 CANCER TREATMENT BY COMBINATION OF EP4 ANTAGONIST AND IMMUNE CHECKPOINT INHIBITOR ONO PHARMACEUTICAL CO., LTD. (JP) 2023-12-07 US disclosed
EP-4252774-A1 COMBINATION THERAPY FOR TREATING PIK3CA-MUTATED CANCER Adlai Nortye Biopharma Co., Ltd. (CN) 2023-10-04 EP disclosed
EP-4245301-A1 CANCER TREATMENT BY COMBINED USE OF EP4 ANTAGONIST AND IMMUNE CHECKPOINT INHIBITOR ONO Pharmaceutical Co., Ltd. (JP) 2023-09-20 EP disclosed
US-11707448-B2 Combination therapies for the treatment of cancer EISAI R&D MANAGEMENT CO., LTD. (JP) 2023-07-25 US disclosed
CN-115697317-A Use of EP4 receptor antagonists for the treatment of liver cancer, melanoma, lymphoma and leukemia 株式会社AskAt 2023-02-03 CN disclosed
WO-2022138793-A1 COMBINATION BETWEEN EP2 RECEPTOR ANTAGONIST AND IMMUNE CHECKPOINT INHIBITOR AND/OR EP4 RECEPTOR ANTAGONIST 小野薬品工業株式会社 2022-06-30 WO disclosed
WO-2022138791-A1 EP2 ANTAGONIST 小野薬品工業株式会社 2022-06-30 WO disclosed
WO-2022111714-A1 COMBINATION THERAPY FOR TREATING PIK3CA-MUTATED CANCER 杭州阿诺生物医药科技有限公司 2022-06-02 WO disclosed
WO-2022102731-A1 CANCER TREATMENT BY COMBINED USE OF EP4 ANTAGONIST AND IMMUNE CHECKPOINT INHIBITOR 小野薬品工業株式会社 2022-05-19 WO disclosed
US-20220071959-A1 COMBINATION THERAPIES FOR THE TREATMENT OF CANCER EISAI R&D MANAGEMENT CO., LTD. (JP) 2022-03-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11707448-B2 Combination therapies for the treatment of cancer PTGER4, PTGER1, PTGER2 PTGER4 1/4885
US-20220071959-A1 COMBINATION THERAPIES FOR THE TREATMENT OF CANCER PTGER4, PTGER1, PTGER2 PTGER4 1/4885
US-20240285640-A1 COMBINATION THERAPY FOR TREATING PIK3CA-MUTATED CANCER PIK3CA, PDPK1, PDCD1 PTGER4 45/4885
US-12240860-B2 Heterobicyclic carboxylic acids and salts thereof PTGER4, PTGER1, GPR4 PTGER4 1/4885
US-20230390303-A1 CANCER TREATMENT BY COMBINATION OF EP4 ANTAGONIST AND IMMUNE CHECKPOINT INHIBITOR CD274, PTGER4, PDCD1 PTGER4 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.