SCHEMBL29433775

SCHEMBL29433775

O=C1CCc2cc3c(cc2N1)OCO3

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 1/20 0.47
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 3/20 0.44
LMNA P02545 2/20 0.44
TSHR P16473 1/20 0.44
NPC1 O15118 1/20 0.44
MAPK13 O15264 1/20 0.44
MAPK12 P53778 1/20 0.44
MAPK11 Q15759 1/20 0.44
MAPK14 Q16539 1/20 0.44
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
PKM P14618 1/20 0.42
KIF11 P52732 3/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
CYP2C9 P11712 3/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
MAPT P10636 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9092910 1.00 CA9 (0.47) CA9KDM4EALDH1A1LMNATSHR
SCHEMBL9834868 0.83 AHR (0.46) KDM4EALDH1A1LMNAADRA2AADRA2B
SCHEMBL31019369 0.76 KDM4E (0.47) KDM4EALDH1A1LMNATSHRPKM
SCHEMBL23671556 0.72 LMNA (0.44) KDM4EALDH1A1LMNATSHRPKM
SCHEMBL12682656 0.71 CYP11B1 (0.56) CA9ALDH1A1NPC1MAPK13MAPK12
SCHEMBL4104017 0.71 CA9 (0.52) CA9KDM4ELMNANPC1MAPK13
SCHEMBL19278654 0.71 CA9 (0.52) CA9NPC1MAPK13MAPK12MAPK11
SCHEMBL852444 0.71 CA9 (0.52) CA9LMNANPC1MAPK13MAPK12
SCHEMBL5568453 0.71 KDM4E (0.58) KDM4EALDH1A1ADRA2AADRA2BADRA2C
SCHEMBL9597670 0.71 CA9 (0.61) CA9ALDH1A1NPC1MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022051388-A2 QUINOLIN-2(1H)-ONE INHIBITORS OF LATE SV40 FACTOR TRUSTEES OF BOSTON UNIVERSITY (US) 2022-03-10 WO disclosed