SCHEMBL29433976

SCHEMBL29433976

NCc1cccc(CO[C@H]2CCOC2)n1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.48
ADORA3 P0DMS8 1/20 0.48
ADORA2B P29275 1/20 0.48
ADORA1 P30542 1/20 0.48
DCPS Q96C86 1/20 0.41
MCHR1 Q99705 1/20 0.34
CXCR4 P61073 1/20 0.33
PDE10A Q9Y233 1/20 0.33
KCNH2 Q12809 1/20 0.33
DRD4 P21917 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
ATF4 P18848 1/20 0.31
GRM4 Q14833 1/20 0.30
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL536780 1.00 ADORA2A (0.48) ADORA2AADORA3ADORA2BADORA1DCPS
SCHEMBL536779 1.00 ADORA2A (0.48) ADORA2AADORA3ADORA2BADORA1DCPS
SCHEMBL1845258 0.87 ADORA2A (0.46) ADORA2AADORA3ADORA2BADORA1DCPS
SCHEMBL1845253 0.87 ADORA2A (0.46) ADORA2AADORA3ADORA2BADORA1DCPS
SCHEMBL20416885 0.86 ADORA2A (0.46) ADORA2AADORA3ADORA2BADORA1DCPS
SCHEMBL18679939 0.86 ADORA2A (0.48) ADORA2AADORA3ADORA2BADORA1DCPS
SCHEMBL22940745 0.86 ADORA2A (0.48) ADORA2AADORA3ADORA2BADORA1DCPS
SCHEMBL22242037 0.86 ADORA2A (0.50) ADORA2AADORA3ADORA2BADORA1DCPS
SCHEMBL536593 0.86 ADORA2A (0.48) ADORA2AADORA3ADORA2BADORA1DCPS
SCHEMBL536592 0.86 ADORA2A (0.48) ADORA2AADORA3ADORA2BADORA1DCPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114276349-B 2-aminopterine derivatives or salts thereof, and preparation method and application thereof 复旦大学 2024-04-09 CN disclosed
CN-114276349-A 2-aminopteridinone derivative or salt thereof, and preparation method and application thereof 复旦大学 2022-04-05 CN disclosed