SCHEMBL29435759

SCHEMBL29435759

c1cc(OC2CCOCC2)ccn1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 8/20 0.48
PDE9A O76083 1/20 0.40
PDE1A P54750 1/20 0.40
DHFR P00374 1/20 0.39
EPHX2 P34913 1/20 0.38
SYK P43405 1/20 0.37
KAT2B Q92831 1/20 0.37
BAZ2B Q9UIF8 1/20 0.37
IKBKB O14920 1/20 0.37
HRH1 P35367 1/20 0.37
GRM5 P41594 1/20 0.37
APP P05067 1/20 0.36
ACACB O00763 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31540092 0.85 HRH1 (0.43) EPHX2IKBKBHRH1
SCHEMBL20400026 0.85 HRH1 (0.43) EPHX2IKBKBHRH1
SCHEMBL28179921 0.81 CYP19A1 (0.44) LRRK2EPHX2IKBKBHRH1
SCHEMBL77615 0.81 PARP10 (0.48) LRRK2EPHX2IKBKBHRH1
SCHEMBL19717281 0.79 HTR2A (0.37) LRRK2PDE9APDE1AEPHX2IKBKB
SCHEMBL13165443 0.79 CYP19A1 (0.46) LRRK2EPHX2HRH1
SCHEMBL16708022 0.79 HRH1 (0.59) PDE9ADHFRSYKKAT2BBAZ2B
SCHEMBL23753940 0.78 CHRNB2 (0.58) LRRK2PDE9AEPHX2
SCHEMBL30471930 0.78 CHRNB2 (0.58) LRRK2PDE9AEPHX2
SCHEMBL3116000 0.78 EPHX2 (0.39) EPHX2IKBKBHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3959207-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES Celgene Corporation (US) 2022-03-02 EP disclosed