SCHEMBL29435883

SCHEMBL29435883

CC(C)(N)c1ccccn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
NOS3 P29474 2/20 0.42
NOS1 P29475 2/20 0.42
NOS2 P35228 2/20 0.42
PI4KA P42356 1/20 0.42
PI4K2B Q8TCG2 1/20 0.42
PI4K2A Q9BTU6 1/20 0.42
PI4KB Q9UBF8 1/20 0.42
CHRM2 P08172 2/20 0.41
KDM4E B2RXH2 3/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
POLB P06746 1/20 0.40
CCR1 P32246 1/20 0.40
CCR5 P51681 1/20 0.40
CCR8 P51685 1/20 0.40
METAP1 P53582 1/20 0.40
BLM P54132 1/20 0.40
HIF1A Q16665 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1114414 1.00 SMN1; SMN2 (0.54) SMN1; SMN2L3MBTL1NOS3NOS1NOS2
Ammonia Solution, Strong SCHEMBL2082802 0.98 SMN1; SMN2 (0.52) SMN1; SMN2L3MBTL1NOS3NOS1NOS2
Hydrochloric Acid SCHEMBL21810899 0.98 SMN1; SMN2 (0.52) SMN1; SMN2L3MBTL1NOS3NOS1NOS2
Hydrochloric Acid SCHEMBL19814625 0.98 SMN1; SMN2 (0.52) SMN1; SMN2L3MBTL1NOS3NOS1NOS2
SCHEMBL1921572 0.86 SMN1; SMN2 (0.54) SMN1; SMN2L3MBTL1NOS3NOS1NOS2
Hydrochloric Acid SCHEMBL15353020 0.84 SMN1; SMN2 (0.52) SMN1; SMN2L3MBTL1NOS3NOS1NOS2
SCHEMBL10442032 0.82 SMN1; SMN2 (0.61) SMN1; SMN2L3MBTL1NOS3NOS1NOS2
SCHEMBL27615166 0.82 SMN1; SMN2 (0.50) SMN1; SMN2L3MBTL1NOS3NOS1NOS2
SCHEMBL6348517 0.81 SMN1; SMN2 (0.54) SMN1; SMN2L3MBTL1NOS3NOS1NOS2
SCHEMBL29080 0.80 SMN1; SMN2 (0.58) SMN1; SMN2L3MBTL1NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4461733-A1 1-AMINOBENZO[4,5]IMIDAZO[1,2-A]PYRAZINE-3-FORMAMIDE COMPOUND, AND PREPARATION THEREFOR AND USE THEREOF Sun Yat-Sen University (CN) 2024-11-13 EP claimed
CN-114276354-A 1-aminobenzo [4,5] imidazo [1,2-a ] pyrazine-3-formamide compound and preparation and application thereof 中山大学 2022-04-05 CN claimed
US-20250092050-A1 1-AMINOBENZO[4,5]IMIDAZO[1,2-A]PYRAZINE-3-FORMAMIDE COMPOUND, AND PREPARATION THEREFOR AND USE THEREOF SUN YAT-SEN UNIVERSITY (CN) 2025-03-20 US disclosed
EP-4461733-A1 1-AMINOBENZO[4,5]IMIDAZO[1,2-A]PYRAZINE-3-FORMAMIDE COMPOUND, AND PREPARATION THEREFOR AND USE THEREOF Sun Yat-Sen University (CN) 2024-11-13 EP disclosed
CN-113072551-B Nitrogen-containing biphenyl derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-08-13 CN disclosed
US-20240067631-A1 PYRAZOLE DERIVATIVES USEFUL AS NAMPT MODULATORS CYTOKINETICS, INC. 2024-02-29 US disclosed
CN-117529476-A Preparation of substituted 1, 2-diamino heterocyclic derivatives and their use as medicaments 亚飞络思制药公司 2024-02-06 CN disclosed
CN-114276354-B 1-aminobenzo [4,5] imidazo [1,2-a ] pyrazine-3-carboxamide compound, preparation and application thereof 中山大学 2023-06-02 CN disclosed
CN-114585625-A Triazolopyrimidines as A2A/A2B inhibitors 因赛特公司 2022-06-03 CN disclosed
CN-114276354-A 1-aminobenzo [4,5] imidazo [1,2-a ] pyrazine-3-formamide compound and preparation and application thereof 中山大学 2022-04-05 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250092050-A1 1-AMINOBENZO[4,5]IMIDAZO[1,2-A]PYRAZINE-3-FORMAMIDE COMPOUND, AND PREPARATION THEREFOR AND USE THEREOF ADORA1, ADORA2A, ADORA2B SMN1; SMN2 4753/4885L3MBTL1 4260/4885NOS3 1580/4885
US-20240067631-A1 PYRAZOLE DERIVATIVES USEFUL AS NAMPT MODULATORS NAMPT, NNT, NAPRT SMN1; SMN2 2574/4885L3MBTL1 3352/4885NOS3 1192/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.