SCHEMBL29439655

SCHEMBL29439655

Cc1nc2cnc(Cl)nc2c(=O)[nH]1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.45
TNKS2 Q9H2K2 1/20 0.42
TYMS P04818 3/20 0.41
ADORA3 P0DMS8 6/20 0.40
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TYRO3 Q06418 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
CDK4 P11802 1/20 0.38
CCND1 P24385 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22716291 1.00 PARP1 (0.45) PARP1TNKS2TYMSADORA3KDM4E
SCHEMBL31330714 0.82 PARP1 (0.44) PARP1TNKS2TYMSADORA3KDM4E
SCHEMBL29656679 0.77 PARP1 (0.40) PARP1TNKS2TYMSADORA3KDM4E
SCHEMBL21514304 0.77 ALDH1A1 (0.47) PARP1TNKS2TYMSADORA3KDM4E
SCHEMBL21514395 0.77 PARP1 (0.40) PARP1TNKS2TYMSADORA3KDM4E
SCHEMBL21514323 0.77 CYP1A2 (0.47) PARP1TNKS2ADORA3KDM4ENPC1
SCHEMBL29656661 0.76 PARP1 (0.39) PARP1TNKS2TYMSADORA3KDM4E
SCHEMBL21514669 0.76 PARP1 (0.39) PARP1TNKS2TYMSADORA3KDM4E
SCHEMBL21514309 0.74 PARP1 (0.38) PARP1TNKS2TYMSADORA3KDM4E
SCHEMBL26644552 0.74 TYRO3 (0.43) PARP1TNKS2TYMSKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118908957-A Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-11-08 CN disclosed
CN-114222737-B Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-07-26 CN disclosed
EP-3976597-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE Janssen Pharmaceutica NV (BE) 2022-04-06 EP disclosed
CN-114222737-A Small molecule inhibitor of NF-kB induced kinase 詹森药业有限公司 2022-03-22 CN disclosed