Arginine

Arginine

SCHEMBL29456

N=C(N)NCCC[C@@H](N)C(=O)O

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

S1PR1S1PR4S1PR5

The experimentally established mechanism targets of Arginine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OTC P00480 1/20 0.56
DDAH1 O94760 4/20 0.51
NOS2 P35228 6/20 0.50
NOS1 P29475 6/20 0.50
NOS3 P29474 5/20 0.50
GSR P00390 1/20 0.48
CYP2C19 P33261 2/20 0.47
CYP1A2 P05177 2/20 0.47
TSHR P16473 2/20 0.47
GLA P06280 1/20 0.47
NFKB1 P19838 1/20 0.47
APEX1 P27695 1/20 0.47
KMT2A Q03164 2/20 0.45
ALOX15 P16050 1/20 0.45
BLM P54132 1/20 0.45
PMP22 Q01453 1/20 0.45
MEN1 O00255 1/20 0.44
ARG2 P78540 4/20 0.44
ARG1 P05089 3/20 0.44
CYP3A4 P08684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Arginine SCHEMBL29778163 1.00 OTC (0.56) OTCDDAH1NOS2NOS1NOS3
Arginine SCHEMBL2411547 1.00 OTC (0.56) OTCDDAH1NOS2NOS1NOS3
Arginine SCHEMBL30361345 1.00 OTC (0.56) OTCDDAH1NOS2NOS1NOS3
Arginine SCHEMBL288132 1.00 OTC (0.56) OTCDDAH1NOS2NOS1NOS3
Arginine SCHEMBL7928810 1.00 OTC (0.56) OTCDDAH1NOS2NOS1NOS3
Arginine SCHEMBL1791 1.00 OTC (0.56) OTCDDAH1NOS2NOS1NOS3
Arginine SCHEMBL28759066 1.00 OTC (0.56) OTCDDAH1NOS2NOS1NOS3
Arginine SCHEMBL31663499 1.00 OTC (0.56) OTCDDAH1NOS2NOS1NOS3
Arginine SCHEMBL1790 1.00 OTC (0.56) OTCDDAH1NOS2NOS1NOS3
Arginine SCHEMBL6374054 1.00 OTC (0.56) OTCDDAH1NOS2NOS1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 14729 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144842-A1 PHARMACEUTICAL COMPOSITION COMPRISING TRYPTOPHAN AND PHYLLOKININ DERIVATIVE FOR USE IN TREATING PSYCHIATRIC AND PSYCHOLOGICAL CONDITIONS TEMPLE OTORONGO LLC (US) 2026-05-28 US claimed
US-12637499-B2 Adrenomedullin analog, method for producing the same, and pharmaceutical use thereof UNIVERSITY OF MIYAZAKI (JP) 2026-05-26 US claimed
CN-122094997-A Aqueous polyurethane coatings for printing applications 2026-05-26 CN claimed
CN-122070294-A Stable vitreous material based on histidine, arginine and glutamic acid amino acids 阵序补丁有限公司 2026-05-19 CN claimed
EP-4735055-A1 UROKINASE-TYPE PLASMINOGEN ACTIVATOR RECEPTOR (UPAR)-PET/CT IN BRAIN TUMOURS Curasight A/S (DK) 2026-05-06 EP claimed
US-12616761-B2 CXCR4-targeting compounds THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2026-05-05 US claimed
US-20260116921-A1 PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR AND THEIR USE TO TREAT INFLAMMATORY DISEASES PROTAGONIST THERAPEUTICS INC (US) 2026-04-30 US claimed
US-20260097023-A1 UNIT ORAL DOSE COMPOSITIONS COMPOSED OF IBUPROFEN OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF AND FAMOTIDINE OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF FOR THE TREATMENT OF ACUTE PAIN AND THE REDUCTION OF THE SEVERITY AND/OR RISK OF HEARTBURN AND/OR UPSET STOMACH SCHABAR RES ASSOCIATES LLC (US) 2026-04-09 US claimed
US-20260098072-A1 METHODS OF STIMULATING APPETITE AND/OR INCREASING BODY WEIGHT USING NON-NATURALLY OCCURRING MELANOCORTIN RECEPTOR ANTAGONIST ANALOGS ENDEVICA BIO INC (US) 2026-04-09 US claimed
EP-4720086-A1 PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR Zealand Pharma A/S (DK) 2026-04-08 EP claimed
US-4127524-A ANALGESIC VETERANS ADMINISTRATION, THE UNITED STATES OF AMERICA AS REPRESENTED BY 1978-11-28 US claimed
US-4127523-A ANALGESIC VETERANS ADMINISTRATION, THE UNITED STATES OF AMERICA AS REPRESENTED BY 1978-11-28 US claimed
US-4127534-A ANALGESIC VETERANS ADMINISTRATION, THE UNITED STATES OF AMERICA AS REPRESENTED BY 1978-11-28 US claimed
US-4127536-A ANALGESIC VETERANS ADMINISTRATION, THE UNITED STATES OF AMERICA AS REPRESENTED BY 1978-11-28 US claimed
US-4127530-A ANALGESIC VETERANS ADMINISTRATION, THE UNITED STATES OF AMERICA AS REPRESENTED BY 1978-11-28 US claimed
US-4127531-A ANALGESIC VETERANS ADMINISTRATION, THE UNITED STATES OF AMERICA AS REPRESENTED BY 1978-11-28 US claimed
US-4127528-A HEXADECAPEPTIDE, ANALGESIC VETERANS ADMINISTRATION, THE UNITED STATES OF AMERICA AS REPRESENTED BY 1978-11-28 US claimed
US-4127538-A ANALGESIC VETERANS ADMINISTRATION, THE UNITED STATES OF AMERICA AS REPRESENTED BY 1978-11-28 US claimed
US-4127533-A ANALGESIC VETERANS ADMINISTRATION, THE UNITED STATES OF AMERICA AS REPRESENTED BY 1978-11-28 US claimed
US-4127539-A ANALGESIC VETERANS ADMINISTRATION, THE UNITED STATES OF AMERICA AS REPRESENTED BY 1978-11-28 US claimed