SCHEMBL29458796

SCHEMBL29458796

CN1CCN(c2ccc(Nc3ncc4c(n3)NC(=O)NC4)cc2C(F)(F)F)CC1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 10/20 0.59
CDK2 P24941 10/20 0.59
CCNA1 P78396 10/20 0.59
CDK4 P11802 5/20 0.57
CCND3 P30281 5/20 0.57
GSK3B P49841 5/20 0.57
PIM1 P11309 4/20 0.57
MTOR P42345 3/20 0.54
AURKA O14965 1/20 0.52
CCNK O75909 1/20 0.52
SLC2A1 P11166 1/20 0.52
CDK12 Q9NYV4 1/20 0.52
BRD4 O60885 2/20 0.52
EGFR P00533 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29458629 0.88 CCNT1 (0.56) CDK4CCND3BRD4EGFR
SCHEMBL29458711 0.87 TNK2 (0.56) CDK2CDK4CCND3AURKASLC2A1
SCHEMBL29458578 0.87 TNK2 (0.56) CDK4CCND3SLC2A1BRD4EGFR
SCHEMBL29458704 0.84 TNK2 (0.61) EGFR
SCHEMBL29458565 0.76 PTK2 (0.49) EGFR
SCHEMBL10098751 0.74 NUAK1 (0.62) CCNA2CDK2CCNA1CDK4CCND3
SCHEMBL16065776 0.74 TNK2 (0.79)
SCHEMBL25068526 0.74 CCNA2 (1.00) CCNA2CDK2CCNA1CDK4CCND3
SCHEMBL29458512 0.74 MAPK7 (0.56) CDK4EGFR
SCHEMBL4154077 0.73 CCNA2 (0.53) CCNA2CDK2CCNA1CDK4CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109836427-B Pyrimidopyrimidinone compounds and application thereof 暨南大学 2022-04-15 CN disclosed