SCHEMBL29463588

SCHEMBL29463588

COC(=O)c1cc(=O)c2ccc(Br)cc2o1

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.70
ABCG2 Q9UNQ0 1/20 0.57
AKR1B1 P15121 4/20 0.53
ALDH1A1 P00352 3/20 0.52
THRB P10828 1/20 0.51
MAPT P10636 4/20 0.46
GAA P10253 1/20 0.46
MAOB P27338 1/20 0.46
SLC2A1 P11166 1/20 0.44
POLB P06746 3/20 0.44
KMT2A Q03164 2/20 0.44
TSHR P16473 1/20 0.44
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TP53 P04637 1/20 0.43
LMNA P02545 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8117167 0.88 KDM4E (0.58) KDM4EABCG2ALDH1A1MAPTGAA
SCHEMBL8119217 0.84 AKR1B1 (0.74) KDM4EAKR1B1ALDH1A1THRBGAA
SCHEMBL4254491 0.84 KDM4E (0.72) KDM4EAKR1B1ALDH1A1THRBMAPT
SCHEMBL8107875 0.82 KDM4E (1.00) KDM4EAKR1B1ALDH1A1MAPTGAA
SCHEMBL9635473 0.82 KDM4E (0.70) KDM4EABCG2AKR1B1ALDH1A1THRB
SCHEMBL18397901 0.81 AKR1B1 (0.69) KDM4EAKR1B1ALDH1A1POLBKMT2A
SCHEMBL3397825 0.80 MAPT (0.68) KDM4EABCG2ALDH1A1MAPTGAA
SCHEMBL29463595 0.80 MAPT (0.68) KDM4EABCG2ALDH1A1MAPTGAA
SCHEMBL13903598 0.80 PIM1 (0.49) KDM4EABCG2ALDH1A1MAPTKMT2A
SCHEMBL29588216 0.80 PIM1 (0.49) KDM4EABCG2ALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022036040-A1 SYNTHESIS OF SMALL MOLECULES INSPIRED BY PHOMOXANTHONE A WORCESTER POLYTECHNIC INSTITUTE (US) 2022-02-17 WO disclosed