SCHEMBL29464261

SCHEMBL29464261

Brc1cccc(-n2ccnc2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.46
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
CYP3A4 P08684 10/20 0.46
CYP1A2 P05177 8/20 0.45
CYP2D6 P10635 8/20 0.45
TDP1 Q9NUW8 6/20 0.45
MAPK1 P28482 4/20 0.45
ALDH1A1 P00352 4/20 0.45
HSD17B10 Q99714 4/20 0.45
LMNA P02545 4/20 0.45
CYP2C19 P33261 7/20 0.44
ALOX15 P16050 5/20 0.44
HPGD P15428 1/20 0.44
HIF1A Q16665 1/20 0.44
CLK4 Q9HAZ1 2/20 0.43
MAPT P10636 2/20 0.43
TP53 P04637 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MEN1 O00255 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2658834 1.00 CYP19A1 (0.46) CYP19A1CYP11B1CYP11B2CYP3A4CYP1A2
SCHEMBL10066877 0.86 CYP3A4 (0.54) CYP19A1CYP11B1CYP11B2CYP3A4CYP1A2
SCHEMBL28614447 0.84 CYP3A4 (0.52) CYP19A1CYP11B1CYP11B2CYP3A4CYP1A2
SCHEMBL16923125 0.81 CYP3A4 (0.48) CYP19A1CYP11B1CYP11B2CYP3A4CYP1A2
SCHEMBL31138265 0.78 CYP3A4 (0.46) CYP19A1CYP11B1CYP11B2CYP3A4CYP1A2
SCHEMBL2643486 0.78 CYP3A4 (0.51) CYP19A1CYP11B1CYP11B2CYP3A4CYP1A2
SCHEMBL13805938 0.78 CYP3A4 (0.51) CYP19A1CYP11B1CYP11B2CYP3A4CYP1A2
SCHEMBL12487845 0.78 LMNA (0.47) CYP19A1CYP11B1CYP11B2CYP3A4CYP1A2
SCHEMBL16265230 0.77 CYP3A4 (0.44) CYP19A1CYP11B1CYP11B2CYP3A4CYP1A2
SCHEMBL30270572 0.74 CYP3A4 (0.53) CYP3A4CYP1A2CYP2D6TDP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114258393-B Heterocyclic compounds having dual inhibitory activity of phosphatidylinositol 3-kinase delta and gamma and medical uses thereof 中国医药研究开发中心有限公司 2024-11-22 CN disclosed
CN-114258393-A Heterocyclic compound with dual phosphatidylinositol 3-kinase delta and gamma inhibitor activity and medical application thereof 中国医药研究开发中心有限公司 2022-03-29 CN disclosed