SCHEMBL29464871

SCHEMBL29464871

Nc1ccc(C(F)(F)F)c(Cl)n1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.46
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
KMT2A Q03164 1/20 0.44
XPO1 O14980 13/20 0.44
ADRB2 P07550 1/20 0.44
BACE1 P56817 3/20 0.40
RPS6KA5 O75582 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1427778 1.00 PIK3CD (0.46) PIK3CDKDM4EALDH1A1KMT2AXPO1
SCHEMBL17826994 0.83 KDM4E (0.39) PIK3CDKDM4EALDH1A1KMT2AXPO1
Succinchlorimide SCHEMBL28310501 0.82 XPO1 (0.43) PIK3CDKDM4EALDH1A1KMT2AXPO1
SCHEMBL29388275 0.82 XPO1 (0.46) PIK3CDALDH1A1XPO1ADRB2RPS6KA5
SCHEMBL855349 0.82 XPO1 (0.46) PIK3CDALDH1A1XPO1ADRB2RPS6KA5
SCHEMBL11010121 0.76 XPO1 (0.45) PIK3CDXPO1ADRB2RPS6KA5
SCHEMBL30285418 0.76 XPO1 (0.45) PIK3CDXPO1ADRB2RPS6KA5
SCHEMBL11272404 0.76 KDM4E (0.46) PIK3CDKDM4EALDH1A1KMT2ABACE1
SCHEMBL24089023 0.74 XPO1 (0.44) PIK3CDXPO1ADRB2RPS6KA5
SCHEMBL7664844 0.74 XPO1 (0.44) KMT2AXPO1ADRB2RPS6KA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025092989-A1 SUBSTITUTED QUINAZOLINE COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMBINATION THEREOF, AND USE THEREOF 泰州红云制药有限公司 2025-05-08 WO disclosed
CN-119462635-A Quinoline derivatives as alpha 4 beta 7 integrin inhibitors 吉利德科学公司 2025-02-18 CN disclosed
CN-118946555-A Compounds having T-structures formed by at least four rings for use in the treatment of cancer and other indications 瑟拉斯有限公司 2024-11-12 CN disclosed
CN-112969687-B Quinoline derivatives as a4 b 7 integrin inhibitors 吉利德科学公司 2024-08-23 CN disclosed
CN-112969700-B Imidazopyridine derivatives as alpha 4 beta 7 integrin inhibitors 吉利德科学公司 2024-08-20 CN disclosed
CN-113015735-B 5-Hydroxy-7-oxabicyclo [2.2.1] heptane-2-carboxamide derivatives for inducing chondrogenesis for the treatment of joint damage 诺华股份有限公司 2024-06-21 CN disclosed
CN-118084870-A Condensed ring compound 豪夫迈·罗氏有限公司 2024-05-28 CN disclosed
CN-118084867-A Condensed ring compound 豪夫迈·罗氏有限公司 2024-05-28 CN disclosed
CN-118084866-A Condensed ring compound 豪夫迈·罗氏有限公司 2024-05-28 CN disclosed
CN-118084868-A Condensed ring compound 豪夫迈·罗氏有限公司 2024-05-28 CN disclosed
EP-4370515-A1 TRICYCLIC COMPOUNDS AS INHIBITORS OF KRAS Incyte Corporation (US) 2024-05-22 EP disclosed
CN-112105419-B Condensed ring compound 豪夫迈·罗氏有限公司 2024-03-29 CN disclosed
CN-112119075-B Condensed ring compound 豪夫迈·罗氏有限公司 2024-03-12 CN disclosed
CN-116867792-A Tetraepoxyazepine compound and use thereof 基因泰克公司 2023-10-10 CN disclosed
WO-2023287896-A1 TRICYCLIC COMPOUNDS AS INHIBITORS OF KRAS INCYTE CORPORATION (US) 2023-01-19 WO disclosed
CN-109641873-B N- (pyridin-2-yl) pyridine-sulfonamide derivatives and their use for the treatment of disease 诺华股份有限公司 2022-03-18 CN disclosed