SCHEMBL29465747

SCHEMBL29465747

CC(F)(F)c1cc(-c2cnc3cn[nH]c3n2)ccc1Cl

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SGK1 O00141 3/20 0.52
GRIN2B Q13224 11/20 0.50
NOTUM Q6P988 2/20 0.44
GRIN1 Q05586 3/20 0.43
KIF20B Q96Q89 1/20 0.40
MAPK1 P28482 1/20 0.39
MAPT P10636 1/20 0.35
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22772817 1.00 SGK1 (0.52) SGK1GRIN2BNOTUMGRIN1KIF20B
SCHEMBL22772840 0.86 SGK1 (0.50) SGK1GRIN2BGRIN1MAPK1
SCHEMBL29465746 0.86 SGK1 (0.50) SGK1GRIN2BGRIN1MAPK1
SCHEMBL29901465 0.79 GRIN2B (0.53) GRIN2BNOTUMGRIN1
SCHEMBL30015184 0.74 GRIN2B (0.48) SGK1GRIN2BMAPK1MAPT
SCHEMBL22772850 0.74 GRIN2B (0.50) SGK1GRIN2BGRIN1
SCHEMBL28689684 0.72 GRIN2B (0.45) GRIN2BNOTUMGRIN1KIF20BCTSS
SCHEMBL22787220 0.69 GRIN2B (0.81) GRIN2B
SCHEMBL30014996 0.69 SGK1 (0.47) SGK1GRIN2BMAPK1
SCHEMBL30014845 0.69 BCHE (0.61) SGK1GRIN2BMAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3983413-A1 SUBSTITUTED PYRAZOLO-PYRAZINES AND THEIR USE AS GLUN2B RECEPTOR MODULATORS Janssen Pharmaceutica NV (BE) 2022-04-20 EP disclosed