SCHEMBL29471995

SCHEMBL29471995

C[Si](C)(C)C#Cc1ccc(-c2ccc(C#C[Si](C)(C)C)nc2)cn1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.40
MCHR1 Q99705 11/20 0.35
ACACB O00763 3/20 0.33
GRM5 P41594 1/20 0.32
CHRM1 P11229 2/20 0.31
HTR2A P28223 2/20 0.31
CYP2D6 P10635 1/20 0.31
SCN10A Q9Y5Y9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22531721 1.00 BACE1 (0.40) BACE1MCHR1ACACBGRM5CHRM1
SCHEMBL2322584 0.89 MCHR1 (0.45) BACE1MCHR1CHRM1HTR2ACYP2D6
SCHEMBL3958689 0.81 CCR1 (0.43) GRM5
SCHEMBL1914210 0.81 GRM5 (0.39) GRM5
SCHEMBL29350657 0.79 ADRA2A (0.37) BACE1GRM5
SCHEMBL19453039 0.79 HCAR2 (0.34) GRM5
SCHEMBL1137069 0.79 ADRA2A (0.37) BACE1GRM5
SCHEMBL3212577 0.79 ADRA2A (0.36) MCHR1GRM5
SCHEMBL3348341 0.79 GRM5 (0.51) BACE1ACACBGRM5
SCHEMBL8973225 0.79 ADRA2A (0.36) BACE1MCHR1GRM5CHRM1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114173772-A Inhibitors of CD40-CD154 binding 托尼克斯医药控股公司 2022-03-11 CN disclosed
EP-3952853-A1 INHIBITORS OF CD40-CD154 BINDING Tonix Pharmaceuticals Holding Corp. (US) 2022-02-16 EP disclosed