(R)Pk-11195

(R)Pk-11195

SCHEMBL29477174

CC[C@@H](C)N([11CH3])C(=O)c1cc2ccccc2c(-c2ccccc2Cl)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSPO P30536 7/20 1.00
MEN1 O00255 2/20 1.00
KMT2A Q03164 2/20 1.00
CYP3A4 P08684 1/20 1.00
CYP2C9 P11712 1/20 1.00
TSHR P16473 1/20 1.00
ALDH1A1 P00352 1/20 1.00
BLM P54132 1/20 1.00
PMP22 Q01453 1/20 1.00
NR1I3 Q14994 1/20 1.00
NPSR1 Q6W5P4 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(R)Pk-11195 SCHEMBL15118334 1.00 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9
(R)Pk-11195 SCHEMBL7685386 1.00 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9
Pk-11195 SCHEMBL117124 1.00 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9
(R)Pk-11195 SCHEMBL29357086 1.00 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9
(R)Pk-11195 SCHEMBL12790424 1.00 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9
Pk-11195 SCHEMBL29354252 1.00 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9
(R)Pk-11195 SCHEMBL3126094 1.00 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9
Pk-11195 SCHEMBL31060347 1.00 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9
SCHEMBL3046732 0.89 TSPO (0.81) TSPOMEN1KMT2ACYP3A4CYP2C9
SCHEMBL3035734 0.89 TSPO (0.81) TSPOMEN1KMT2ACYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250268847-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF DEMYELINATING DISORDERS THE UNIVERSITY OF CHICAGO (US) 2025-08-28 US disclosed
US-12310933-B2 Treatment of demyelinating disorders THE UNIVERSITY OF CHICAGO (US) 2025-05-27 US disclosed
WO-2025068949-A1 EMRUSOLMIN FOR USE IN TREATING MULTIPLE SYSTEM ATROPHY TEVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2025-04-03 WO disclosed
CN-118344351-A Preparation method and application of PET imaging agent targeting neuroinflammatory purinergic P2Y12 receptor 复旦大学 2024-07-16 CN disclosed
US-20240009332-A1 COMPOSITE EMBOLIZATION BEADS TRANSLATIONAL AND FUNDAMENTAL TECHNOLOGIES INSTITUTE LLC 2024-01-11 US disclosed
US-20230322897-A1 COMPOSITIONS AND METHODS FOR TREATING NEUROCOGNITIVE DISORDERS AVROBIO, INC. 2023-10-12 US disclosed
US-20230243811-A1 IDENTIFICATION OF TRANSPLANTED HUMAN CELLS RIGSHOSPITALET (REGH) (DK) 2023-08-03 US disclosed
US-11712487-B2 Composite embolization beads RAIKA MEDICAL IMAGING INC. (US) 2023-08-01 US disclosed
US-11672468-B2 System and method for multi-modality quantification of neuroinflammation in central nervous system diseases WASHINGTON UNIVERSITY (US) 2023-06-13 US disclosed
EP-4175717-A2 COMPOSITIONS AND METHODS FOR TREATING NEUROCOGNITIVE DISORDERS Avrobio, Inc. (US) 2023-05-10 EP disclosed
US-20220133850-A1 COMPOSITIONS AND METHODS FOR TREATING NEUROCOGNITIVE DISORDERS AVROBIO, INC. 2022-05-05 US disclosed
US-20220111005-A1 COMPOSITIONS AND METHODS FOR TREATING NEUROCOGNITIVE DISORDERS AVROBIO, INC. (US) 2022-04-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250268847-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF DEMYELINATING DISORDERS MAG, PMP22, GBA1 TSPO 2564/4885MEN1 3520/4885KMT2A 2511/4885
US-12310933-B2 Treatment of demyelinating disorders MAG, PMP22, GBA1 TSPO 1892/4885MEN1 3454/4885KMT2A 2239/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.