SCHEMBL29478802

SCHEMBL29478802

Cc1ccc(F)c(C(C)O)c1Br

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
EPAS1 Q99814 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24373240 1.00 MEN1 (0.32) MEN1KMT2AHDAC1HDAC6EPAS1
SCHEMBL30662731 0.85 MEN1 (0.34) MEN1KMT2AEPAS1
SCHEMBL22331229 0.85 MEN1 (0.34) MEN1KMT2AEPAS1
SCHEMBL20872550 0.79 CHRM2 (0.34) MEN1KMT2A
SCHEMBL29628557 0.79 CHRM2 (0.34) MEN1KMT2A
SCHEMBL3093413 0.79 MEN1 (0.33) MEN1KMT2A
SCHEMBL25015121 0.76 MEN1 (0.32) MEN1KMT2A
SCHEMBL3097748 0.76 CHRM2 (0.32) MEN1KMT2A
SCHEMBL13069751 0.75 DAO (0.33) MEN1KMT2A
SCHEMBL10324344 0.73 MEN1 (0.33) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4232444-A1 HETEROCYCLIC SPIRO COMPOUNDS AND METHODS OF USE Amgen Inc. (US) 2023-08-30 EP disclosed
WO-2022083569-A1 HETEROCYCLIC SPIRO COMPOUNDS AND METHODS OF USE AMGEN INC. (US) 2022-04-28 WO disclosed