SCHEMBL29480760

SCHEMBL29480760

COC(c1ccc(Br)nc1)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 2/20 0.32
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
DGAT1 O75907 1/20 0.30
CHRNB2 P17787 1/20 0.30
CHRNA4 P43681 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12281762 1.00 CYP26A1 (0.32) CYP26A1NR1H2NR1H3DGAT1CHRNB2
SCHEMBL12282137 0.83 NR3C1 (0.38)
SCHEMBL12283943 0.81 CYP2D6 (0.33) NR1H2NR1H3
SCHEMBL12199222 0.81 CYP2D6 (0.33) NR1H2NR1H3
SCHEMBL12199391 0.81 CYP2D6 (0.33) NR1H2NR1H3
SCHEMBL12199465 0.79 AKR1C3 (0.35) DGAT1CHRNB2CHRNA4
SCHEMBL12200016 0.79 AKR1C3 (0.35) DGAT1CHRNB2CHRNA4
SCHEMBL12181540 0.77 KRAS (0.34) NR1H2NR1H3
SCHEMBL31292671 0.77 DEGS1 (0.38)
SCHEMBL31463701 0.77 DEGS1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114174294-A Novel compounds for inhibiting JANUS kinase 1 人类制药有限公司 2022-03-11 CN disclosed