SCHEMBL2948452

SCHEMBL2948452

O=C(O)Cc1c(Cl)nc(Cc2ccc(NC(=O)C=Cc3ccccc3)cc2)n2ccnc12

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 4/20 0.51
RAB9A P51151 2/20 0.46
NPC1 O15118 1/20 0.46
EGFR P00533 7/20 0.45
MMP1 P03956 5/20 0.45
MMP2 P08253 5/20 0.45
MMP9 P14780 5/20 0.45
HPSE Q9Y251 1/20 0.44
DHFR P00374 3/20 0.42
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
DEGS1 O15121 1/20 0.41
NAMPT P43490 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2948450 1.00 PTGDR2 (0.51) PTGDR2RAB9ANPC1EGFRMMP1
SCHEMBL2946922 0.94 PTGDR2 (0.54) PTGDR2RAB9ANPC1EGFRMMP1
SCHEMBL2946919 0.94 PTGDR2 (0.54) PTGDR2RAB9ANPC1EGFRMMP1
SCHEMBL2942672 0.80 NR1H4 (0.55) PTGDR2RAB9ANPC1
SCHEMBL2948543 0.78 KDM4E (0.55) PTGDR2RAB9ANPC1
SCHEMBL2942781 0.78 PTGDR2 (0.36) PTGDR2
SCHEMBL2941686 0.77 PTGDR2 (0.56) PTGDR2
SCHEMBL5959181 0.77 MAPT (0.44) PTGDR2RAB9ANPC1EGFRMMP1
SCHEMBL1652116 0.76 PTGDR2 (0.54) PTGDR2RAB9AEGFRMMP1MMP2
SCHEMBL1652115 0.76 PTGDR2 (0.54) PTGDR2RAB9AEGFRMMP1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7750014-B2 Imidazo[1,2-C]pyrimidinylacetic acid derivatives ACTIMIS PHARMACEUTICALS, INC. (US) 2010-07-06 US claimed
EP-1718649-B1 IMIDAZO 1,2-C PYRIMIDINYLACETIC ACID DERIVATIVES ACTIMIS PHARMACEUTICALS INC (US) 2009-06-10 EP claimed
US-20090012102-A1 Imidazo[1,2-C]Pyrimidinylacetic Acid Derivatives ACTIMIS PHARMACEUTICALS, INC. (US) 2009-01-08 US claimed
EP-1718649-A2 IMIDAZO 1,2-C PYRIMIDINYLACETIC ACID DERIVATIVES Actimis Pharmaceuticals, Inc., (US) 2006-11-08 EP claimed
WO-2005073234-A2 IMIDAZO[1,2-C]PYRIMIDINYLACETIC ACID DERIVATIVES ACTIMIS PHARMACEUTICALS, INC. (US) 2005-08-11 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090012102-A1 Imidazo[1,2-C]Pyrimidinylacetic Acid Derivatives HRH2, CCR2, HRH1 PTGDR2 56/4885RAB9A 1284/4885NPC1 2986/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.