SCHEMBL29484607

SCHEMBL29484607

CC(C)(C)OC(=O)NC1CCN(C(=O)c2ccnc(Nc3ccccc3)n2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.50
CFTR P13569 2/20 0.49
CKS1B P61024 1/20 0.49
SKP1 P63208 1/20 0.49
SKP2 Q13309 1/20 0.49
PARP1 P09874 3/20 0.47
KCNA3 P22001 1/20 0.43
AKT1 P31749 1/20 0.43
ADORA2A P29274 2/20 0.43
ADORA2B P29275 2/20 0.43
MERTK Q12866 1/20 0.42
EPHX2 P34913 1/20 0.42
NPC1L1 Q9UHC9 1/20 0.42
KDM1A O60341 1/20 0.41
MAOB P27338 1/20 0.41
DRD2 P14416 1/20 0.41
CCNT1 O60563 1/20 0.41
CCNA2 P20248 1/20 0.41
CDK2 P24941 1/20 0.41
CDK9 P50750 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29484598 1.00 NAMPT (0.50) NAMPTCFTRCKS1BSKP1SKP2
SCHEMBL25882312 1.00 NAMPT (0.50) NAMPTCFTRCKS1BSKP1SKP2
SCHEMBL30471161 0.86 ALDH1A1 (0.42) ADORA2BCCNT1CCNA2CDK2CDK9
SCHEMBL25311631 0.86 EPHX2 (0.48) EPHX2CDK2
SCHEMBL25879044 0.85 EPHX2 (0.47) EPHX2CCNA2CDK2CCNA1
SCHEMBL25883636 0.84 NAMPT (0.52) NAMPTCFTRCKS1BSKP1SKP2
SCHEMBL30471249 0.84 NAMPT (0.52) NAMPTCFTRCKS1BSKP1SKP2
SCHEMBL29466333 0.84 CCNA2 (0.54) CFTRCKS1BSKP1SKP2CCNT1
SCHEMBL25882559 0.84 CCNA2 (0.54) CFTRCKS1BSKP1SKP2CCNT1
SCHEMBL29466335 0.80 GSK3A (0.50) CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022057932-A1 CARBONYL HETEROCYCLIC COMPOUND AND APPLICATION THEREOF 上海医药集团股份有限公司 2022-03-24 WO disclosed
WO-2022057928-A1 CARBONYL HETEROCYCLIC COMPOUND AND APPLICATION THEREOF 上海医药集团股份有限公司 2022-03-24 WO disclosed