SCHEMBL2949189

SCHEMBL2949189

Cc1cccc(C)c1-c1nc(Nc2ccc(N3CCNCC3)cc2)nc2c1c(N)nn2CCCN1CCCCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNK2 Q07912 4/20 0.46
STK17A Q9UEE5 1/20 0.41
CDK4 P11802 12/20 0.40
CCND1 P24385 9/20 0.40
CCND2 P30279 6/20 0.40
CCND3 P30281 6/20 0.40
FGFR1 P11362 4/20 0.40
FGFR2 P21802 4/20 0.40
FGFR4 P22455 4/20 0.40
FGFR3 P22607 4/20 0.40
CCNA2 P20248 4/20 0.40
CDK2 P24941 4/20 0.40
NUAK1 O60285 1/20 0.40
CCNB2 O95067 1/20 0.40
CCNE2 O96020 1/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
CCNE1 P24864 1/20 0.40
CCNA1 P78396 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2957977 0.93 TNK2 (0.46) TNK2CDK4CCND1CCND2CCND3
SCHEMBL2953623 0.88 TNK2 (0.57) TNK2FGFR1CCNA2CDK2CCNA1
SCHEMBL2959696 0.87 TNK2 (0.58) TNK2FGFR1SRC
SCHEMBL2952193 0.85 TNK2 (0.64) TNK2STK17ACDK4CCND1CCND2
SCHEMBL2952192 0.81 TNK2 (0.47) TNK2CDK4CCND1CCND3CCNA2
SCHEMBL30338613 0.77 TNK2 (0.77) TNK2
SCHEMBL2956900 0.76 TNK2 (0.58) TNK2SRC
SCHEMBL2956876 0.73 TNK2 (0.69) TNK2SRC
SCHEMBL2955951 0.73 TNK2 (0.42) TNK2SRC
SCHEMBL2957964 0.73 TNK2 (0.50) TNK2SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7763624-B2 Substituted pyrazolo[3,4-d]pyrimidines as ACK-1 and LCK inhibitors AMGEN INC. (US) 2010-07-27 US claimed
US-20070072851-A1 Pyrazolopyridine and pyrazolopyrimidine compounds AMGEN INC. (US) 2007-03-29 US claimed
US-7763624-B2 Substituted pyrazolo[3,4-d]pyrimidines as ACK-1 and LCK inhibitors AMGEN INC. (US) 2010-07-27 US disclosed
US-20070072851-A1 Pyrazolopyridine and pyrazolopyrimidine compounds AMGEN INC. (US) 2007-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070072851-A1 Pyrazolopyridine and pyrazolopyrimidine compounds LCK, MAP4K5, TPMT TNK2 113/4885STK17A 94/4885CDK4 200/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.