SCHEMBL2956900

SCHEMBL2956900

Cc1cccc(C)c1-c1nc(Nc2ccccc2)nc2c1c(N)nn2CCN1CCOCC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNK2 Q07912 4/20 0.58
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
RAB9A P51151 1/20 0.46
ILK Q13418 1/20 0.43
SRC P12931 2/20 0.43
MAPK1 P28482 2/20 0.42
HTT P42858 2/20 0.42
ALDH1A1 P00352 3/20 0.41
MAPT P10636 3/20 0.41
ALOX15 P16050 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP3A4 P08684 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
KDR P35968 1/20 0.41
FLT3 P36888 1/20 0.41
LMNA P02545 2/20 0.41
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2952192 0.89 TNK2 (0.47) TNK2SRCMAPK1MAPTFLT3
SCHEMBL2959696 0.86 TNK2 (0.58) TNK2SRCKDM4ECYP3A4KDR
SCHEMBL2955937 0.86 SRC (0.52) TNK2SRCMAPTCYP3A4HPGD
SCHEMBL2953623 0.86 TNK2 (0.57) TNK2SRCKDM4ECYP3A4KDR
SCHEMBL2955951 0.81 TNK2 (0.42) TNK2SRCIGF1RCA12CA2
SCHEMBL2957977 0.77 TNK2 (0.46) TNK2SRCKDRFLT3IGF1R
SCHEMBL4701225 0.77 TNK2 (0.49) TNK2MEN1KMT2ARAB9ASRC
SCHEMBL2949189 0.76 TNK2 (0.46) TNK2SRC
SCHEMBL30338760 0.74 TNK2 (1.00) TNK2KDR
SCHEMBL2952193 0.72 TNK2 (0.64) TNK2KDRWEE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7763624-B2 Substituted pyrazolo[3,4-d]pyrimidines as ACK-1 and LCK inhibitors AMGEN INC. (US) 2010-07-27 US claimed
US-20070072851-A1 Pyrazolopyridine and pyrazolopyrimidine compounds AMGEN INC. (US) 2007-03-29 US claimed
US-7763624-B2 Substituted pyrazolo[3,4-d]pyrimidines as ACK-1 and LCK inhibitors AMGEN INC. (US) 2010-07-27 US disclosed
US-20070072851-A1 Pyrazolopyridine and pyrazolopyrimidine compounds AMGEN INC. (US) 2007-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070072851-A1 Pyrazolopyridine and pyrazolopyrimidine compounds LCK, MAP4K5, TPMT TNK2 113/4885MEN1 1368/4885KMT2A 2887/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.