SCHEMBL29496151

SCHEMBL29496151

CCc1ccc(-c2c(F)ccc3cc(Cl)cnc23)c(N)n1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.35
USP7 Q93009 3/20 0.33
BACE1 P56817 7/20 0.32
BACE2 Q9Y5Z0 2/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
CTSD P07339 3/20 0.31
CNR1 P21554 1/20 0.31
CCR1 P32246 1/20 0.30
CCR5 P51681 1/20 0.30
CCR8 P51685 1/20 0.30
FGFR2 P21802 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29496187 0.89 FGFR1 (0.35) USP7PTGS1PTGS2CCR1CCR5
SCHEMBL29496138 0.89 USP7 (0.33) PDE10AUSP7CCR1CCR5CCR8
Hydrochloric Acid SCHEMBL29496160 0.87 BACE1 (0.33) PDE10AUSP7BACE1BACE2CYP3A4
SCHEMBL29496143 0.87 PDPK1 (0.34) USP7BACE1BACE2CTSD
SCHEMBL29496273 0.86 USP7 (0.32) USP7BACE1PTGS1PTGS2CTSD
SCHEMBL24671049 0.83 FGFR1 (0.35) BACE1BACE2CYP3A4CYP2D6CTSD
SCHEMBL29495873 0.83 FGFR1 (0.35) BACE1BACE2CYP3A4CYP2D6CTSD
SCHEMBL29496209 0.82 FGFR1 (0.32) USP7
SCHEMBL22969595 0.81 REN (0.39) PDE10AUSP7BACE1BACE2CYP3A4
SCHEMBL29495834 0.81 REN (0.39) PDE10AUSP7BACE1BACE2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114269730-A 5-heteroaryl-pyridin-2-amine compounds as neuropeptide FF receptor antagonists 多曼治疗学公司 2022-04-01 CN disclosed