Acitretin

Acitretin

SCHEMBL29496318

COc1cc(C)c(/C=C/C(C)=C/C=C/C(C)=C/C(=O)O)c(C)c1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

RARARARBRARGRXRARXRBRXRG

The experimentally established mechanism targets of Acitretin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA known ✓ P19793 12/20 0.45
RARG known ✓ P13631 9/20 0.45
RARA known ✓ P10276 6/20 0.45
RARB known ✓ P10826 6/20 0.45
RXRB known ✓ P28702 4/20 0.45
RXRG known ✓ P48443 4/20 0.45
ALDH1A1 P00352 8/20 1.00
MAPT P10636 7/20 1.00
SMN1; SMN2 Q16637 4/20 1.00
ABCB11 O95342 2/20 1.00
ABCC4 O15439 1/20 1.00
NR1I2 O75469 1/20 1.00
PTGS1 P23219 4/20 0.72
ADORA3 P0DMS8 3/20 0.72
PGR P06401 2/20 0.72
CHRM1 P11229 2/20 0.72
SLC6A2 P23975 2/20 0.72
ESR1 P03372 1/20 0.72
SLC6A4 P31645 1/20 0.72
OPRM1 P35372 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acitretin SCHEMBL159360 1.00 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2ABCB11ABCC4
Acitretin SCHEMBL29883491 1.00 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2ABCB11ABCC4
Acitretin SCHEMBL5028866 1.00 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2ABCB11ABCC4
Acitretin SCHEMBL3759 1.00 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2ABCB11ABCC4
Acitretin SCHEMBL2280089 1.00 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2ABCB11ABCC4
Acitretin SCHEMBL5053805 1.00 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2ABCB11ABCC4
Acitretin SCHEMBL10750446 0.99 ALDH1A1 (0.98) ALDH1A1MAPTSMN1; SMN2ABCB11ABCC4
Acitretin SCHEMBL4443721 0.99 ALDH1A1 (0.98) ALDH1A1MAPTSMN1; SMN2ABCB11ABCC4
Acitretin SCHEMBL9856594 0.94 ALDH1A1 (0.89) ALDH1A1MAPTSMN1; SMN2ABCB11ABCC4
SCHEMBL10750080 0.94 ALDH1A1 (0.89) ALDH1A1MAPTSMN1; SMN2ABCB11ABCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119394085-A Real-time monitoring method and system for characteristics of cooling tower of wet cooling unit 上海明华电力科技有限公司 2025-02-07 CN claimed
US-20240420847-A1 SYSTEM AND METHODS FOR PERFORMING SALIVA-BASED DIAGNOSTIC SCREENINGS CellectGen, Inc. (US) 2024-12-19 US claimed
WO-2024174011-A1 LIPOSOME, METHOD FOR PREPARING A LIPOSOME, INTRANASAL COMPOSITION COMPRISING A LIPOSOME, METHOD FOR PREPARING AN INTRANASAL COMPOSITION, KIT AND USE OF THE COMPOSITION ROSSI BERGMANN BARTIRA (BR) 2024-08-29 WO claimed
CN-116510024-A Composition, preparation method and application thereof 上海复东生物医药有限责任公司 2023-08-01 CN claimed
WO-2023133084-A1 SYSTEM AND METHODS FOR PERFORMING SALIVA-BASED DIAGNOSTIC SCREENINGS CellectGen, Inc. (US) 2023-07-13 WO claimed
US-12521358-B2 Method for selecting cancer patients for whom combination therapy with retinoid and cancer therapeutic agent is effective, and combination medicament with retinoid and cancer therapeutic agent RAQUALIA PHARMA INC. (JP) 2026-01-13 US disclosed
US-20250172609-A1 PROBE TESTING APPARATUS, PROBE TESTING SYSTEM AND PROBE CARD RENESAS ELECTRONICS CORPORATION (JP) 2025-05-29 US disclosed
CN-120044280-A Probe testing device, probe testing system and probe card 瑞萨电子株式会社 2025-05-27 CN disclosed
CN-119603433-A Projector automatic focusing method based on gradient calculation and convolution neural network 佛山得一智能科技有限公司 2025-03-11 CN disclosed
US-20240420847-A1 SYSTEM AND METHODS FOR PERFORMING SALIVA-BASED DIAGNOSTIC SCREENINGS CellectGen, Inc. (US) 2024-12-19 US disclosed
US-20240317815-A1 T-CELL MODULATORY MULTIMERIC POLYPEPTIDES AND METHODS OF USE THEREOF CUE BIOPHARMA INC (US) 2024-09-26 US disclosed
WO-2024174011-A1 LIPOSOME, METHOD FOR PREPARING A LIPOSOME, INTRANASAL COMPOSITION COMPRISING A LIPOSOME, METHOD FOR PREPARING AN INTRANASAL COMPOSITION, KIT AND USE OF THE COMPOSITION ROSSI BERGMANN BARTIRA (BR) 2024-08-29 WO disclosed
WO-2023133084-A1 SYSTEM AND METHODS FOR PERFORMING SALIVA-BASED DIAGNOSTIC SCREENINGS CellectGen, Inc. (US) 2023-07-13 WO disclosed
EP-3495349-B1 (HETERO)ARYL CYCLOPROPYLAMINE COMPOUNDS AS LSD1 INHIBITORS ORYZON GENOMICS SA (ES) 2023-06-28 EP disclosed
EP-3498297-B1 PHARMACEUTICAL COMPOSITION FOR THE TREATMENT OF AUTISM STALICLA S A (CH) 2023-06-21 EP disclosed
EP-4173639-A1 METHOD FOR SELECTING CANCER PATIENT FOR WHICH COMBINATION THERAPY OF RETINOID AND CANCER TREATMENT AGENT WILL BE EFFECTIVE, AND COMBINED DRUG OF RETINOID AND CANCER TREATMENT AGENT RaQualia Pharma Inc. (JP) 2023-05-03 EP disclosed
CN-115634198-A Solvent composition for water-insoluble substances and preparation method and application thereof 浙江贝灵生物医药有限公司 2023-01-24 CN disclosed
EP-4074695-A1 (HETERO)ARYL CYCLOPROPYLAMINE COMPOUNDS AS LSD1 INHIBITORS Oryzon Genomics, S.A. (ES) 2022-10-19 EP disclosed
US-11439627-B2 Pharmaceutical composition for the treatment of autism Stalicla S.A. (CH) 2022-09-13 US disclosed
EP-3984555-A1 PHARMACEUTICAL COMPOSITION FOR THE TREATMENT OF AUTISM Stalicla S.A. (CH) 2022-04-20 EP disclosed