SCHEMBL29501322

SCHEMBL29501322

O=Cc1cc(NC2CCOCC2)ncn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 7/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
MAP2K7 O14733 1/20 0.41
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
ALOX15 P16050 1/20 0.39
CYP2C19 P33261 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
LRRK2 Q5S007 1/20 0.38
CDK2 P24941 5/20 0.38
CCNE1 P24864 4/20 0.38
MAPK3 P27361 3/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25389374 1.00 MAPK1 (0.42) MAPK1MEN1KMT2AMAP2K7CYP1A2
SCHEMBL28629361 0.91 MEN1 (0.37) MAPK1MEN1KMT2AMAP2K7CYP1A2
SCHEMBL29501387 0.84 MEN1 (0.37) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL28999535 0.84 MEN1 (0.37) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL29501437 0.82 CYP1A2 (0.49) MAPK1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL28883687 0.82 CYP1A2 (0.49) MAPK1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL28999380 0.79 HRH4 (0.46) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL28999356 0.79 MEN1 (0.40) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL15229185 0.76 MEN1 (0.71) MAPK1MEN1KMT2AMAP2K7CYP1A2
SCHEMBL15830049 0.76 MAPK1 (0.50) MAPK1MEN1KMT2AMAP2K7CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116113626-A Compound with anti-tumor activity and application thereof 上海翊石医药科技有限公司 2023-05-12 CN disclosed
WO-2022048631-A1 COMPOUND HAVING ANTITUMOR ACTIVITY AND USE THEREOF 上海翊石医药科技有限公司 2022-03-10 WO disclosed