SCHEMBL29501437

SCHEMBL29501437

O=Cc1cc(NC2CCNCC2)ncn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.49
HSD17B10 Q99714 3/20 0.49
CYP3A4 P08684 2/20 0.49
ALOX15 P16050 2/20 0.49
CYP2C19 P33261 2/20 0.49
ALDH1A1 P00352 2/20 0.49
CYP2C9 P11712 1/20 0.49
MAPK1 P28482 1/20 0.46
HRH3 Q9Y5N1 3/20 0.44
HRH4 Q9H3N8 3/20 0.44
HRH2 P25021 1/20 0.44
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
AURKA O14965 1/20 0.36
RPS6KB1 P23443 1/20 0.36
CYP2D6 P10635 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
PRMT5 O14744 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28883687 1.00 CYP1A2 (0.49) CYP1A2HSD17B10CYP3A4ALOX15CYP2C19
SCHEMBL29501322 0.82 MAPK1 (0.42) CYP1A2HSD17B10CYP3A4ALOX15CYP2C19
SCHEMBL25389374 0.82 MAPK1 (0.42) CYP1A2HSD17B10CYP3A4ALOX15CYP2C19
SCHEMBL28999356 0.79 MEN1 (0.40) CYP1A2HSD17B10CYP3A4ALOX15CYP2C19
SCHEMBL28999380 0.79 HRH4 (0.46) CYP1A2HSD17B10CYP3A4ALOX15CYP2C19
SCHEMBL29501387 0.78 MEN1 (0.37) CYP1A2HSD17B10CYP3A4ALOX15CYP2C19
SCHEMBL28999535 0.78 MEN1 (0.37) CYP1A2HSD17B10CYP3A4ALOX15CYP2C19
SCHEMBL28629361 0.77 MEN1 (0.37) CYP1A2HSD17B10CYP3A4ALOX15CYP2C19
SCHEMBL2349988 0.76 CYP1A2 (0.59) CYP1A2HSD17B10CYP3A4ALOX15CYP2C19
SCHEMBL21139461 0.76 CYP1A2 (0.56) CYP1A2HSD17B10CYP3A4ALOX15CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116113626-A Compound with anti-tumor activity and application thereof 上海翊石医药科技有限公司 2023-05-12 CN disclosed
WO-2022048631-A1 COMPOUND HAVING ANTITUMOR ACTIVITY AND USE THEREOF 上海翊石医药科技有限公司 2022-03-10 WO disclosed