SCHEMBL29501356

SCHEMBL29501356

Clc1ccc(Nc2cc(N3CCC(N4CCc5ccccc5C4)CC3)ncn2)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.48
CHRM4 P08173 5/20 0.46
CHRM2 P08172 1/20 0.46
CHRM5 P08912 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
CXCR3 P49682 1/20 0.45
PRCP P42785 1/20 0.41
ADRA1A P35348 4/20 0.40
HRH4 Q9H3N8 1/20 0.40
ABL1 P00519 1/20 0.39
BCR P11274 1/20 0.39
SMO Q99835 1/20 0.39
EGFR P00533 1/20 0.38
ERBB3 P21860 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26248126 0.92 SCN9A (0.53) SCN9ACHRM4CHRM2CHRM5CHRM1
SCHEMBL26248321 0.91 SCN9A (0.51) SCN9ACHRM4CHRM1ADRA1AHRH4
SCHEMBL29501484 0.91 SCN9A (0.51) SCN9ACHRM4CHRM1ADRA1AHRH4
SCHEMBL26248334 0.90 SCN9A (0.53) SCN9ACHRM4CHRM2CHRM5CHRM1
SCHEMBL29501463 0.90 SCN9A (0.53) SCN9ACHRM4CHRM2CHRM5CHRM1
SCHEMBL29501346 0.90 SCN9A (0.48) SCN9ACHRM4CHRM2CHRM5CHRM1
SCHEMBL26248210 0.90 SCN9A (0.48) SCN9ACHRM4CHRM2CHRM5CHRM1
SCHEMBL29501379 0.89 SCN9A (0.47) SCN9ACHRM4CHRM2CHRM5CHRM1
SCHEMBL26248283 0.89 SCN9A (0.47) SCN9ACHRM4CHRM2CHRM5CHRM1
SCHEMBL26248494 0.89 SCN9A (0.48) SCN9ACHRM4CHRM2CHRM5CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022048631-A1 COMPOUND HAVING ANTITUMOR ACTIVITY AND USE THEREOF 上海翊石医药科技有限公司 2022-03-10 WO disclosed