SCHEMBL29501475

SCHEMBL29501475

c1ccc2c(c1)CCN(C1CCN(c3cc(NC4CCC4)ncn3)CC1)C2

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.52
DPP4 P27487 3/20 0.43
SMO Q99835 1/20 0.42
ADRA1A P35348 4/20 0.42
SCN9A Q15858 1/20 0.41
PRMT5 O14744 4/20 0.41
WDR77 Q9BQA1 4/20 0.41
CHRM4 P08173 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26248522 0.97 HRH4 (0.51) HRH4DPP4SMOADRA1ASCN9A
SCHEMBL26254464 0.91 HRH4 (0.49) HRH4DPP4SMOADRA1ASCN9A
SCHEMBL26254803 0.90 HRH4 (0.50) HRH4DPP4SMOADRA1ASCN9A
SCHEMBL29501378 0.90 HRH4 (0.50) HRH4DPP4SMOADRA1ASCN9A
SCHEMBL26248111 0.86 PRMT5 (0.54) HRH4ADRA1ASCN9APRMT5WDR77
SCHEMBL25387542 0.85 PRMT5 (0.50) HRH4DPP4SCN9APRMT5WDR77
SCHEMBL26254679 0.85 PRMT5 (0.50) HRH4DPP4SCN9APRMT5WDR77
SCHEMBL25387544 0.85 PRMT5 (0.50) HRH4DPP4SCN9APRMT5WDR77
SCHEMBL26248126 0.84 SCN9A (0.53) HRH4SMOADRA1ASCN9ACHRM4
SCHEMBL29501410 0.82 SCN9A (0.50) HRH4SMOADRA1ASCN9ACHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022048631-A1 COMPOUND HAVING ANTITUMOR ACTIVITY AND USE THEREOF 上海翊石医药科技有限公司 2022-03-10 WO disclosed