SCHEMBL2950866

SCHEMBL2950866

NC(c1ccncc1)c1ccc2ncc(-c3cc4ccccc4o3)n2n1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 20/20 0.60
FYN P06241 1/20 0.60
MKNK2 Q9HBH9 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2940427 0.87 MKNK1 (0.60) MKNK1FYNMKNK2
SCHEMBL2945059 0.79 FYN (0.45) MKNK1FYNMKNK2
SCHEMBL14771339 0.79 MKNK1 (0.74) MKNK1FYNMKNK2
SCHEMBL15921290 0.78 MKNK1 (0.73) MKNK1FYNMKNK2
SCHEMBL2949526 0.77 PIK3CD (0.52) MKNK1FYNMKNK2
SCHEMBL13859054 0.76 MKNK1 (1.00) MKNK1FYNMKNK2
SCHEMBL19336870 0.76 MKNK1 (0.73) MKNK1MKNK2
SCHEMBL30521685 0.75 MKNK1 (1.00) MKNK1FYN
SCHEMBL2950870 0.75 MKNK1 (1.00) MKNK1FYN
SCHEMBL14764375 0.75 MKNK1 (0.64) MKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7750000-B2 Substituted imidazo[1,2b]pyridazines as kinase inhibitors, their preparation and use as medicaments BAYER SCHERING PHARMA AG (DE) 2010-07-06 US disclosed
US-20070093490-A1 Substituted imidazo[1,2b]pyridazines as kinase inhibitors, their preparation and use as medicaments BAYER INTELLECTUAL PROPERTY GMBH (DE) 2007-04-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070093490-A1 Substituted imidazo[1,2b]pyridazines as kinase inhibitors, their preparation and use as medicaments MAP4K2, MAP3K1, MAP3K2 MKNK1 144/4885FYN 421/4885MKNK2 79/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.