SCHEMBL29520545

SCHEMBL29520545

CC(C)=C1C(c2ccccc2)=NC(C(C)(C)C)=Nc2ccc(C)cc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.42
RAB9A P51151 5/20 0.42
NPC1 O15118 4/20 0.42
LMNA P02545 2/20 0.35
CHRM1 P11229 2/20 0.34
KMT2A Q03164 6/20 0.33
MEN1 O00255 5/20 0.33
SMN1; SMN2 Q16637 4/20 0.33
KDM4E B2RXH2 3/20 0.33
TP53 P04637 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
CDK5 Q00535 1/20 0.33
CDK5R1 Q15078 1/20 0.33
TDP1 Q9NUW8 2/20 0.33
PKM P14618 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
CYP3A4 P08684 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29409248 0.91 NPC1 (0.36) MAPTRAB9ANPC1LMNACHRM1
SCHEMBL29520576 0.86 IDO1 (0.31) IDO1
SCHEMBL29520664 0.86 CHRM1 (0.39) MAPTLMNACHRM1KMT2AMEN1
SCHEMBL29521036 0.86 CYP2C9 (0.36) MAPTRAB9ANPC1LMNACHRM1
SCHEMBL29520721 0.84 MEN1 (0.33) MAPTRAB9ANPC1LMNAKMT2A
SCHEMBL29520828 0.84 MAPT (0.45) MAPTRAB9ANPC1LMNAKMT2A
SCHEMBL29520554 0.84 CHRM1 (0.37) CHRM1
SCHEMBL28500399 0.84 MAPT (0.43) MAPTNPC1LMNACHRM1KMT2A
SCHEMBL29520292 0.84 CNR1 (0.35) MAPTRAB9ANPC1LMNAKMT2A
SCHEMBL29520737 0.83 IDO1 (0.40) MAPTLMNAKMT2AMEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112174901-B Synthesis method and anticancer activity of 1, 3-benzodiazepine compound 河南师范大学 2022-02-08 CN disclosed