SCHEMBL29520758

SCHEMBL29520758

N[C@@H](CO)C(=O)NCCc1ccc(O)c(O)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.61
HSD17B10 Q99714 4/20 0.59
MAPT P10636 4/20 0.59
HIF1A Q16665 3/20 0.59
KDM4E B2RXH2 3/20 0.59
PTGS1 P23219 2/20 0.59
ALDH1A1 P00352 2/20 0.59
LMNA P02545 2/20 0.59
HPGD P15428 2/20 0.59
BLM P54132 2/20 0.59
SLC7A5 Q01650 3/20 0.53
ERCC1 P07992 1/20 0.52
ERCC4 Q92889 1/20 0.52
CA1 P00915 2/20 0.51
CA2 P00918 2/20 0.51
CA9 Q16790 2/20 0.51
CA7 P43166 1/20 0.51
CA14 Q9ULX7 1/20 0.51
APP P05067 1/20 0.50
GLI1 P08151 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24277517 1.00 HDAC8 (0.61) HDAC8HSD17B10MAPTHIF1AKDM4E
SCHEMBL24277516 1.00 HDAC8 (0.61) HDAC8HSD17B10MAPTHIF1AKDM4E
SCHEMBL15399610 0.88 HDAC8 (0.61) HDAC8HSD17B10MAPTHIF1AKDM4E
SCHEMBL3690574 0.87 HDAC8 (0.60) HDAC8HSD17B10MAPTHIF1AKDM4E
SCHEMBL26980197 0.87 HDAC8 (0.60) HDAC8HSD17B10MAPTHIF1AKDM4E
SCHEMBL26305770 0.86 HDAC8 (0.59) HDAC8HSD17B10MAPTHIF1AKDM4E
SCHEMBL24277699 0.85 HDAC8 (0.45) HDAC8HSD17B10MAPTHIF1AKDM4E
SCHEMBL24277700 0.85 HDAC8 (0.45) HDAC8HSD17B10MAPTHIF1AKDM4E
SCHEMBL28976207 0.85 MAPT (0.58) HDAC8HSD17B10MAPTHIF1AKDM4E
SCHEMBL7559848 0.85 HDAC8 (0.64) HDAC8HSD17B10MAPTHIF1AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4211114-A1 SMALL MOLECULE INHIBITORS OF ENPP1 The Regents of the University of California (US) 2023-07-19 EP disclosed
WO-2022056068-A1 SMALL MOLECULE INHIBITORS OF ENPP1 THE REGENTS OF THE UNIVERSITY OFCALIFORNIA (US) 2022-03-17 WO disclosed