SCHEMBL7559848

SCHEMBL7559848

N[C@@H](Cc1ccc(O)cc1)C(=O)NCCc1ccc(O)c(O)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.64
SLC7A5 Q01650 4/20 0.59
KDM4E B2RXH2 2/20 0.58
PTGS1 P23219 2/20 0.58
HIF1A Q16665 2/20 0.58
HSD17B10 Q99714 2/20 0.58
LMNA P02545 2/20 0.58
ALDH1A1 P00352 1/20 0.58
MAPT P10636 1/20 0.58
HPGD P15428 1/20 0.58
BLM P54132 1/20 0.58
YARS1 P54577 2/20 0.57
BCHE P06276 1/20 0.54
ACHE P22303 1/20 0.54
EGFR P00533 2/20 0.52
LCK P06239 2/20 0.52
FYN P06241 2/20 0.52
ADORA3 P0DMS8 2/20 0.52
HTR2A P28223 2/20 0.52
PTGS2 P35354 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11753174 0.91 SLC7A5 (0.63) HDAC8SLC7A5KDM4EPTGS1HIF1A
SCHEMBL20865641 0.89 HDAC8 (0.64) HDAC8SLC7A5KDM4E
Hydrochloric Acid SCHEMBL20854816 0.87 HDAC8 (0.67) HDAC8SLC7A5KDM4E
SCHEMBL24277516 0.85 HDAC8 (0.61) HDAC8SLC7A5KDM4EPTGS1HIF1A
SCHEMBL29520758 0.85 HDAC8 (0.61) HDAC8SLC7A5KDM4EPTGS1HIF1A
SCHEMBL24277517 0.85 HDAC8 (0.61) HDAC8SLC7A5KDM4EPTGS1HIF1A
SCHEMBL15399610 0.85 HDAC8 (0.61) HDAC8SLC7A5KDM4EPTGS1HIF1A
SCHEMBL3690574 0.83 HDAC8 (0.60) HDAC8SLC7A5KDM4EPTGS1HIF1A
SCHEMBL29220965 0.83 HDAC8 (0.59) HDAC8SLC7A5KDM4ECA1CA2
SCHEMBL26980197 0.83 HDAC8 (0.60) HDAC8SLC7A5KDM4EPTGS1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165492-A1 HYDROXYPHENYL DERIVATIVES WITH HIV INTEGRASE INHIBITORY PROPERTIES Pharmacor Inc. (CA) 2002-01-02 EP disclosed
WO-2000059867-A1 HYDROXYPHENYL DERIVATIVES WITH HIV INTEGRASE INHIBITORY PROPERTIES PHARMACOR INC. (CA) 2000-10-12 WO disclosed
US-4033997-A Preparation of dopamine derivatives ABBOTT LABORATORIES (US) 1977-07-05 US disclosed