SCHEMBL29520778

SCHEMBL29520778

CC(C)=C1C(c2ccccc2)=NC(C(C)(C)C)=Nc2cc(Cl)ccc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 3/20 0.37
OPRK1 P41145 3/20 0.36
LMNA P02545 2/20 0.36
PDE3A Q14432 1/20 0.36
CCNE2 O96020 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
TP53 P04637 2/20 0.34
RXFP1 Q9HBX9 1/20 0.34
HSD11B1 P28845 1/20 0.34
RPS6KA3 P51812 1/20 0.34
NR1I2 O75469 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
HTR2C P28335 1/20 0.34
ADRA1A P35348 1/20 0.34
PTGS2 P35354 1/20 0.34
CHRNA4 P43681 1/20 0.34
SLC6A3 Q01959 1/20 0.34
PDE4D Q08499 1/20 0.34
SHMT1 P34896 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29520664 0.91 CHRM1 (0.39) CHRM1OPRK1LMNAPDE3ACCNE2
SCHEMBL29520739 0.86 CNR1 (0.34) PTGS2SLC6A3NPC1ALDH1A1HPGD
SCHEMBL29409248 0.86 NPC1 (0.36) CHRM1LMNATP53RXFP1MEN1
SCHEMBL29520620 0.85 CNR1 (0.38) KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL29520737 0.83 IDO1 (0.40) LMNAMEN1KMT2AALDH1A1HPGD
SCHEMBL29520545 0.80 MAPT (0.42) CHRM1LMNATP53MEN1KMT2A
SCHEMBL29520576 0.79 IDO1 (0.31)
SCHEMBL29521036 0.79 CYP2C9 (0.36) CHRM1LMNATP53MEN1KMT2A
SCHEMBL29520641 0.77 CYP2A6 (0.33) HSD11B1
SCHEMBL29520721 0.76 MEN1 (0.33) LMNAMEN1KMT2ANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112174901-B Synthesis method and anticancer activity of 1, 3-benzodiazepine compound 河南师范大学 2022-02-08 CN disclosed