SCHEMBL2952147

SCHEMBL2952147

COC(=O)c1ccc(-c2ccc(Cl)nc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 1/20 0.50
KCNQ3 O43525 1/20 0.49
KCNQ2 O43526 1/20 0.49
CA1 P00915 4/20 0.49
CA2 P00918 4/20 0.49
CA12 O43570 3/20 0.49
CA9 Q16790 3/20 0.49
CA14 Q9ULX7 3/20 0.49
MAPK1 P28482 2/20 0.49
NAPRT Q6XQN6 1/20 0.49
RHEB Q15382 1/20 0.48
TDP1 Q9NUW8 1/20 0.47
CA7 P43166 1/20 0.47
SGK1 O00141 1/20 0.47
CAMKK2 Q96RR4 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MKNK1 Q9BUB5 1/20 0.46
MKNK2 Q9HBH9 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38659193 1.00 KDM4E (0.50) KDM4EALDH1A1KCNQ3KCNQ2CA1
SCHEMBL29552438 0.86 MAPK1 (0.65) KDM4EALDH1A1MAPK1NAPRTTDP1
SCHEMBL64640 0.86 MAPK1 (0.65) KDM4EALDH1A1MAPK1NAPRTTDP1
SCHEMBL20241211 0.84 MAPK1 (0.62) KDM4EALDH1A1MAPK1NAPRTTDP1
SCHEMBL29776105 0.84 MAPK1 (0.62) KDM4EALDH1A1MAPK1NAPRTTDP1
SCHEMBL17687665 0.83 KDM4E (0.53) KDM4EALDH1A1CA1CA2CA12
SCHEMBL38656713 0.83 CA12 (0.52) KDM4EALDH1A1KCNQ3KCNQ2CA1
SCHEMBL2943965 0.81 CA1 (0.53) KDM4EALDH1A1CA1CA2CA12
SCHEMBL22392835 0.81 KCNQ3 (0.46) KDM4EALDH1A1KCNQ3KCNQ2RHEB
SCHEMBL30421160 0.81 KCNQ3 (0.46) KDM4EALDH1A1KCNQ3KCNQ2RHEB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026102082-A1 ALKYLPHENYL SUBSTITUTED COMPOUNDS, COMPOSITIONS AND METHODS OF USE DEEP APPLE THERAPEUTICS, INC. (US) 2026-05-15 WO disclosed
US-20260132119-A1 Alkylphenyl Substituted Compounds, Compositions and Methods of Use DEEP APPLE THERAPEUTICS, INC. (US) 2026-05-14 US disclosed
US-7754886-B2 N-acylsulfonamide apoptosis promoters ABBOTT LABORATORIES (US) 2010-07-13 US disclosed
US-20090137585-A1 N-ACYLSULFONAMIDE APOPTOSIS PROMOTERS ABBOTT LABORATORIES (US) 2009-05-28 US disclosed
US-7504512-B2 N-acylsulfonamide apoptosis promoters ABBOTT LABORATORIES (US) 2009-03-17 US disclosed
EP-1318978-B1 N-ACYLSULFONAMIDE APOPTOSIS PROMOTERS ABBOTT LAB (US) 2006-02-08 EP disclosed
US-20040192681-A1 N-acylsulfonamide apoptosis promoters ABBVIE INC. 2004-09-30 US disclosed
US-6720338-B2 BCL-X1 INHIBITING COMPOSITIONS AND METHODS OF PROMOTING APOPTOSIS IN A MAMMAL ABBOTT LABORATORIES 2004-04-13 US disclosed
EP-1318978-A2 N-ACYLSULFONAMIDE APOPTOSIS PROMOTERS Abbott Laboratories (US) 2003-06-18 EP disclosed
US-20020086887-A1 N-Acylsulfonamide apoptosis promoters ABBVIE INC. 2002-07-04 US disclosed
US-20020055631-A1 N-acylsulfonamide apoptosis promoters ABBOTT LABORATORIES 2002-05-09 US disclosed
WO-2002024636-A2 N-ACYLSULFONAMIDE APOPTOSIS PROMOTERS ABBOTT LABORATORIES (US) 2002-03-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020086887-A1 N-Acylsulfonamide apoptosis promoters BAX, BCLAF1, BCL2 KDM4E 1911/4885ALDH1A1 2651/4885KCNQ3 4474/4885
US-20020055631-A1 N-acylsulfonamide apoptosis promoters BAX, BCLAF1, BCL2 KDM4E 1563/4885ALDH1A1 2460/4885KCNQ3 4538/4885
US-20040192681-A1 N-acylsulfonamide apoptosis promoters BAX, BCLAF1, BCL2 KDM4E 1911/4885ALDH1A1 2651/4885KCNQ3 4474/4885
US-20090137585-A1 N-ACYLSULFONAMIDE APOPTOSIS PROMOTERS BAX, BCL2, BCOR KDM4E 1143/4885ALDH1A1 3404/4885KCNQ3 4439/4885
US-20260132119-A1 Alkylphenyl Substituted Compounds, Compositions and Methods of Use GIPR, MC2R, GRPR KDM4E 3829/4885ALDH1A1 3360/4885KCNQ3 2562/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.