SCHEMBL29530751

SCHEMBL29530751

NC(=O)Cc1csc(NC(c2ccccc2)(c2ccccc2)c2ccccc2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 1/20 0.50
PDE5A O76074 6/20 0.46
KDM4E B2RXH2 2/20 0.46
GAA P10253 3/20 0.45
MAPT P10636 3/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
TP53 P04637 2/20 0.42
LMNA P02545 1/20 0.42
PDE1A P54750 2/20 0.41
PDE1B Q01064 2/20 0.41
PDE1C Q14123 2/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2786872 0.89 GAA (0.53) PDE5AKDM4EGAAMAPTMEN1
SCHEMBL11091142 0.86 PDE5A (0.46) PDE5AKDM4EGAAMAPTMEN1
SCHEMBL10756603 0.86 PDE5A (0.46) PDE5AKDM4EGAAMAPTMEN1
SCHEMBL2786880 0.84 TP53 (0.59) GAAMAPTMEN1KMT2AALDH1A1
SCHEMBL27481508 0.83 PDE5A (0.43) PDE5AKDM4EGAAMAPTMEN1
SCHEMBL10464685 0.82 PDE5A (0.41) PDE5AKDM4EGAAMAPTMEN1
SCHEMBL17596693 0.80 SCD (0.41) PDE5AKDM4EGAAMAPTMEN1
SCHEMBL6584892 0.80 SMN1; SMN2 (0.45) PDE5AKDM4EGAAMAPTMEN1
SCHEMBL27815401 0.79 NPC1 (0.51) KDM4EMAPTMEN1KMT2AALDH1A1
SCHEMBL10437870 0.79 PDE5A (0.39) PDE5AKDM4EGAAMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114213433-B Process for the preparation of C-3 tetrahydrofuran substituted cephalosporin-siderophore conjugates 重庆医药高等专科学校 2023-03-24 CN disclosed
CN-114213433-A Process for the preparation of C-3 tetrahydrofuran substituted cephalosporin-siderophore conjugates 重庆医药高等专科学校 2022-03-22 CN disclosed