SCHEMBL295393

SCHEMBL295393

CCCCCOc1c(Br)cc(CCC(C)(N)CO)cc1Br

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
THRA P10827 4/20 0.55
THRB P10828 4/20 0.55
S1PR1 P21453 10/20 0.44
S1PR3 Q99500 8/20 0.44
S1PR4 O95977 7/20 0.44
S1PR5 Q9H228 6/20 0.44
S1PR2 O95136 1/20 0.43
LPAR2 Q9HBW0 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
TNNC1 P63316 5/20 0.40
SGPL1 O95470 1/20 0.40
GPR183 P32249 1/20 0.40
CERS2 Q96G23 1/20 0.40
SPHK2 Q9NRA0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL295392 1.00 THRA (0.55) THRATHRBS1PR1S1PR3S1PR4
Hydrochloric Acid SCHEMBL295255 0.99 THRA (0.54) THRATHRBS1PR1S1PR3S1PR4
Hydrochloric Acid SCHEMBL295254 0.99 THRA (0.54) THRATHRBS1PR1S1PR3S1PR4
SCHEMBL295364 0.93 THRA (0.48) THRATHRBS1PR1S1PR3S1PR4
SCHEMBL295363 0.93 THRA (0.48) THRATHRBS1PR1S1PR3S1PR4
SCHEMBL294681 0.87 SMN1; SMN2 (0.46) THRATHRBS1PR1S1PR3S1PR4
SCHEMBL294682 0.87 SMN1; SMN2 (0.46) THRATHRBS1PR1S1PR3S1PR4
SCHEMBL365503 0.85 S1PR1 (0.45) THRATHRBS1PR1S1PR3S1PR4
SCHEMBL294540 0.82 SMN1; SMN2 (0.42) THRATHRBS1PR1S1PR3S1PR4
SCHEMBL294539 0.82 SMN1; SMN2 (0.42) THRATHRBS1PR1S1PR3S1PR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636171-B1 AMINO-PROPANOL DERIVATIVES AS SPHINGOSINE-1-PHOSPHATE RECEPTOR MODULATORS NOVARTIS AG (CH) 2012-03-14 EP claimed