SCHEMBL29540558

SCHEMBL29540558

Fc1ccc(-c2ccn(-c3ccnc4[nH]ccc34)n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.48
CSNK1D P48730 2/20 0.48
MAPK11 Q15759 1/20 0.48
PRKCI P41743 4/20 0.46
MAPK1 P28482 1/20 0.44
EGFR P00533 3/20 0.41
AKT2 P31751 1/20 0.40
NUDT1 P36639 5/20 0.38
AXL P30530 1/20 0.38
IKBKB O14920 1/20 0.38
CHUK O15111 1/20 0.38
DAPK3 O43293 1/20 0.38
JAK2 O60674 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38
PAK4 O96013 1/20 0.38
CSF1R P07333 1/20 0.38
RET P07949 1/20 0.38
IGF1R P08069 1/20 0.38
FGFR1 P11362 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL100645 1.00 MAPK14 (0.48) MAPK14CSNK1DMAPK11PRKCIMAPK1
Trifluoroacetic Acid SCHEMBL4092178 0.90 MAPK14 (0.41) MAPK14CSNK1DMAPK11PRKCIMAPK1
SCHEMBL29540449 0.87 PRKCI (0.46) MAPK14CSNK1DMAPK11PRKCIAKT2
SCHEMBL28055281 0.87 PRKCI (0.46) PRKCIMAPK1AKT2NUDT1AXL
SCHEMBL102456 0.87 PRKCI (0.46) MAPK14CSNK1DMAPK11PRKCIAKT2
SCHEMBL100939 0.87 JAK2 (0.52) PRKCIMAPK1AKT2NUDT1IKBKB
SCHEMBL29540619 0.87 JAK2 (0.52) PRKCIMAPK1AKT2NUDT1IKBKB
SCHEMBL100644 0.84 MAPK1 (0.47) PRKCIMAPK1AKT2ROCK1
SCHEMBL29540798 0.84 MAPK1 (0.47) PRKCIMAPK1AKT2ROCK1
SCHEMBL99492 0.84 PRKCI (0.43) PRKCIAKT2NUDT1AXLIKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11744832-B2 Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors INCYTE CORPORATION (US) 2023-09-05 US disclosed
US-20220395506-A1 HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS INCYTE CORPORATION 2022-12-15 US disclosed
US-11331320-B2 Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors INCYTE HOLDINGS CORPORATION (US) 2022-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220395506-A1 HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS JAK3, JAK1, JAK2 MAPK14 362/4885CSNK1D 1611/4885MAPK11 550/4885
US-11744832-B2 Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors JAK3, JAK1, JAK2 MAPK14 362/4885CSNK1D 1611/4885MAPK11 550/4885
US-11331320-B2 Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors JAK3, JAK1, JAK2 MAPK14 362/4885CSNK1D 1611/4885MAPK11 550/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.