SCHEMBL29544972

SCHEMBL29544972

COc1c(Cl)cccc1Nc1c(-c2ccnc3ccncc23)nn2c1C(=O)NCC2

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.37
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
TYK2 P29597 7/20 0.34
PIK3CA P42336 1/20 0.32
MTOR P42345 1/20 0.32
PARP1 P09874 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29544407 0.89 CCNT1 (0.34) EGFRCCNT1CDK9TYK2PARP1
SCHEMBL29544554 0.88 BRD4 (0.38) EGFRCCNT1CDK9TYK2
SCHEMBL29544735 0.88 CCNT1 (0.34) EGFRCCNT1CDK9TYK2PIK3CA
SCHEMBL29544781 0.88 CCNT1 (0.34) EGFRCCNT1CDK9TYK2PIK3CA
SCHEMBL29545142 0.87 CSF1R (0.39) EGFRCCNT1CDK9TYK2
SCHEMBL29544730 0.87 EGFR (0.42) EGFRTYK2
SCHEMBL29544438 0.86 TYK2 (0.36) EGFRCCNT1CDK9TYK2PARP1
SCHEMBL29544599 0.85 EGFR (0.36) EGFRCCNT1CDK9TYK2
SCHEMBL29545092 0.85 EGFR (0.39) EGFRCCNT1CDK9TYK2
SCHEMBL29544958 0.85 TYK2 (0.34) EGFRCCNT1CDK9TYK2PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022072634-A1 BICYCLIC COMPOUNDS FOR USE IN THE TREATMENT CANCER SCORPION THERAPEUTICS, INC. (US) 2022-04-07 WO disclosed