SCHEMBL29545140

SCHEMBL29545140

COc1c(F)cccc1Nc1c(-c2ccnc3cn[nH]c23)nn2c1C(=O)NCC2

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.42
TYK2 P29597 8/20 0.35
ROCK2 O75116 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C8 P10632 2/20 0.34
TGFBR1 P36897 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29544438 0.91 TYK2 (0.36) EGFRTYK2CYP3A4CYP2C8TGFBR1
SCHEMBL29545012 0.87 EGFR (0.41) EGFRTYK2ROCK2
SCHEMBL29544468 0.85 EGFR (0.41) EGFRTYK2ROCK2
SCHEMBL29544703 0.84 EGFR (0.38) EGFRTYK2ROCK2CYP3A4CYP2C8
SCHEMBL29544852 0.84 EGFR (0.49) EGFRROCK2
SCHEMBL29544860 0.84 EGFR (0.49) EGFRROCK2
SCHEMBL29544736 0.83 EGFR (0.40) EGFRTYK2
SCHEMBL29544418 0.83 EGFR (0.39) EGFRTYK2CYP3A4CYP2C8TGFBR1
SCHEMBL29544775 0.82 EGFR (0.47) EGFRROCK2
SCHEMBL29545225 0.82 EGFR (0.47) EGFRTYK2ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022072634-A1 BICYCLIC COMPOUNDS FOR USE IN THE TREATMENT CANCER SCORPION THERAPEUTICS, INC. (US) 2022-04-07 WO disclosed