SCHEMBL29548628

SCHEMBL29548628

CC(C)(C)OC(=O)N1C[C@@H](NC(=O)c2ccc(NC(=O)c3ccccc3)cc2)C[C@H]1C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 7/20 0.52
USP30 Q70CQ3 2/20 0.45
ANPEP P15144 4/20 0.44
NPC1 O15118 4/20 0.44
NR1H2 P55055 1/20 0.44
CACNA1B Q00975 1/20 0.41
APBA1 Q02410 1/20 0.41
KDM4E B2RXH2 2/20 0.41
PKM P14618 1/20 0.41
RAB9A P51151 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
POLB P06746 1/20 0.40
PTPN1 P18031 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2707643 0.93 MMP2 (0.59) MMP2USP30ANPEPNR1H2KDM4E
SCHEMBL2709145 0.93 MMP2 (0.59) MMP2USP30ANPEPNR1H2KDM4E
SCHEMBL29548256 0.92 MMP2 (0.64) MMP2USP30ANPEPNPC1NR1H2
SCHEMBL29548777 0.91 MMP2 (0.49) MMP2USP30ANPEPNPC1NR1H2
SCHEMBL12609045 0.90 MMP2 (0.52) MMP2USP30ANPEPNPC1NR1H2
SCHEMBL29548395 0.89 USP30 (0.57) MMP2USP30ANPEPNPC1NR1H2
SCHEMBL29548707 0.86 NR1H2 (0.42) MMP2NPC1NR1H2KDM4EPKM
SCHEMBL3110842 0.84 MMP2 (0.73) MMP2USP30ANPEPNR1H2KDM4E
SCHEMBL6365330 0.84 MMP2 (0.73) MMP2USP30ANPEPNR1H2KDM4E
SCHEMBL3110836 0.84 MMP2 (0.73) MMP2USP30ANPEPNR1H2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022087630-A1 INHIBITORS OF AMINO ACID TRANSPORT ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2022-04-28 WO disclosed