SCHEMBL29549573

SCHEMBL29549573

Nc1ncc(-c2cnn(CCO)c2)c2scc(-c3ccc4c(C(=O)Nc5ccccc5)cccc4c3)c12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 12/20 1.00
BTK Q06187 10/20 0.66
FGFR1 P11362 7/20 0.66
AURKB Q96GD4 6/20 0.66
FER P16591 5/20 0.66
BLK P51451 5/20 0.66
STK3 Q13188 5/20 0.66
RET P07949 5/20 0.66
PDGFRA P16234 5/20 0.66
AURKA O14965 5/20 0.66
RPS6KA3 P51812 5/20 0.66
MAP4K4 O95819 5/20 0.66
NTRK1 P04629 5/20 0.66
FYN P06241 5/20 0.66
MET P08581 5/20 0.66
NTRK3 Q16288 5/20 0.66
NTRK2 Q16620 5/20 0.66
TAOK1 Q7L7X3 5/20 0.66
FLT1 P17948 5/20 0.66
KIT P10721 5/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17034027 1.00 KDR (1.00) KDRBTKFGFR1AURKBFER
SCHEMBL18579380 0.87 KDR (0.76) KDRBTKFGFR1AURKBFER
Ilorasertib SCHEMBL3381224 0.79 KDR (1.00) KDRBTKFGFR1AURKBFER
Ilorasertib SCHEMBL29373142 0.79 KDR (1.00) KDRBTKFGFR1AURKBFER
Ilorasertib SCHEMBL29496449 0.79 KDR (1.00) KDRBTKFGFR1AURKBFER
SCHEMBL5472344 0.79 KDR (0.65) KDRBTKFGFR1AURKBFER
Ilorasertib SCHEMBL30406133 0.79 KDR (0.98) KDRBTKFGFR1AURKBFER
Ilorasertib SCHEMBL11898929 0.79 KDR (0.98) KDRBTKFGFR1AURKBFER
Ilorasertib SCHEMBL11900182 0.79 KDR (0.94) KDRBTKFGFR1AURKBFER
Ilorasertib SCHEMBL11899788 0.79 KDR (0.94) KDRBTKFGFR1AURKBFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3112351-B1 NAPHTHYLAMIDE COMPOUND, PREPARATION METHOD AND USE THEREOF SHANGHAI INST MATERIA MEDICA CAS (CN) 2022-03-30 EP disclosed