SCHEMBL29554697

SCHEMBL29554697

CC(=O)c1cc2cccc(Cl)c2nc1-c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.50
SMO Q99835 3/20 0.39
CNR2 P34972 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
PARP1 P09874 2/20 0.39
PPARA Q07869 1/20 0.39
POLB P06746 2/20 0.38
THRB P10828 1/20 0.38
RORB Q92753 1/20 0.38
TP53 P04637 1/20 0.38
HSD11B1 P28845 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CYP1A2 P05177 2/20 0.37
PTPN1 P18031 1/20 0.37
PTGS2 P35354 1/20 0.37
LMNA P02545 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KDM4E B2RXH2 1/20 0.37
CA12 O43570 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4191610 0.80 MAOB (0.40) RXFP1PARP1POLBCYP1A2PTPN1
SCHEMBL16597147 0.77 PDE10A (0.57) DHODHPOLBCYP1A2LMNACYP2C9
SCHEMBL19413117 0.77 DHODH (0.46) DHODHTP53KDM4E
SCHEMBL19646360 0.77 DHODH (0.43) DHODHRXFP1POLBTHRBTP53
SCHEMBL457871 0.75 DHODH (0.44) DHODHRXFP1NPSR1CYP1A2PTGS2
SCHEMBL29617462 0.74 DHODH (0.44) DHODHTP53LMNAKDM4E
SCHEMBL27802982 0.74 DHODH (0.43) DHODHTHRBLMNAKDM4E
SCHEMBL1880602 0.74 DHODH (0.46) DHODHTP53NPSR1CYP1A2CYP2C9
SCHEMBL9958654 0.72 DHODH (0.49) DHODHHSD11B1CYP1A2LMNAKDM4E
SCHEMBL26617907 0.72 KEAP1 (0.47) RXFP1TP53LMNAKDM4ECA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109516974-B Preparation method of substituted pyrimidine PI3K inhibitor 南京圣和药业股份有限公司 2022-05-27 CN disclosed