SCHEMBL29558358

SCHEMBL29558358

Clc1ccc(CNc2nc3ccccc3nc2Nc2ccc(Cl)c(Cl)c2)cc1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 1/20 0.49
USP1 O94782 1/20 0.47
WDR48 Q8TAF3 1/20 0.47
SLC2A1 P11166 1/20 0.46
MEN1 O00255 2/20 0.46
POLB P06746 2/20 0.46
KMT2A Q03164 2/20 0.46
TYMS P04818 1/20 0.44
ADORA3 P0DMS8 4/20 0.44
HTR2B P41595 1/20 0.43
TMEM97 Q5BJF2 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
CHEK1 O14757 1/20 0.42
ROCK2 O75116 1/20 0.42
RPS6KA5 O75582 1/20 0.42
MAP4K4 O95819 1/20 0.42
CHEK2 O96017 1/20 0.42
PIM1 P11309 1/20 0.42
PRKACA P17612 1/20 0.42
RPS6KB1 P23443 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29558270 0.92 APP (0.48) NPY5RSLC2A1MEN1POLBKMT2A
SCHEMBL29559170 0.90 ABCG2 (0.44) NPY5RUSP1WDR48SLC2A1MEN1
SCHEMBL28725367 0.83 USP1 (0.51) USP1WDR48KMT2ARPS6KB1DYRK1A
SCHEMBL29558289 0.83 USP1 (0.51) USP1WDR48KMT2ARPS6KB1DYRK1A
SCHEMBL29558591 0.82 HRH4 (0.41) NPY5RUSP1WDR48MEN1KMT2A
SCHEMBL29559166 0.81 SOS1 (0.59) MEN1POLBKMT2AMAPK1ALDH1A1
SCHEMBL29559492 0.80 FLT1 (0.56) NPY5RMEN1POLBKMT2AMAPK1
SCHEMBL29558650 0.79 CTNNB1 (0.46) MEN1POLBKMT2AALDH1A1MAPT
SCHEMBL29558870 0.78 APP (0.47) LMNAHTT
SCHEMBL29559506 0.77 MEN1 (0.59) MEN1KMT2AMAPK1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114380753-A Aryl or heteroaryl substituted quinoxaline-2, 3-diamine compound and antibacterial application thereof 中国医学科学院药物研究所 2022-04-22 CN claimed
CN-114380753-A Aryl or heteroaryl substituted quinoxaline-2, 3-diamine compound and antibacterial application thereof 中国医学科学院药物研究所 2022-04-22 CN disclosed