SCHEMBL29558644

SCHEMBL29558644

Fc1cc(Nc2nc3ccccc3nc2NCc2ccco2)cc(F)c1F

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.55
ALDH1A1 P00352 7/20 0.53
TSHR P16473 4/20 0.53
POLB P06746 3/20 0.53
USP2 O75604 1/20 0.53
SOS1 Q07889 4/20 0.52
KMT2A Q03164 8/20 0.51
MAPT P10636 8/20 0.51
MEN1 O00255 7/20 0.51
MAPK1 P28482 4/20 0.51
NPSR1 Q6W5P4 3/20 0.51
XBP1 P17861 1/20 0.51
HSD17B10 Q99714 4/20 0.49
HTT P42858 3/20 0.49
HPGD P15428 2/20 0.49
LMNA P02545 2/20 0.49
GAA P10253 1/20 0.49
TP53 P04637 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
CASP1 P29466 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29558247 0.80 KDM4E (0.66) KDM4EALDH1A1TSHRPOLBUSP2
SCHEMBL29559166 0.80 SOS1 (0.59) KDM4EALDH1A1TSHRPOLBUSP2
SCHEMBL29558517 0.79 KDM4E (0.49) KDM4EPOLBKMT2AMAPTMEN1
SCHEMBL29558521 0.78 NTRK1 (0.45) KDM4EALDH1A1POLBKMT2AMAPT
SCHEMBL29558367 0.77 APP (0.47) KMT2AMAPTLMNATP53SMN1; SMN2
SCHEMBL28725385 0.73 KDM4E (0.60) KDM4EALDH1A1TSHRPOLBUSP2
SCHEMBL29558895 0.73 KDM4E (0.60) KDM4EALDH1A1TSHRPOLBUSP2
SCHEMBL29558251 0.68 MAPT (0.49) KDM4EPOLBKMT2AMAPTMEN1
SCHEMBL1084254 0.68 KMT2A (1.00) KDM4EALDH1A1TSHRPOLBSOS1
SCHEMBL4356051 0.67 ALDH1A1 (0.49) KDM4EALDH1A1TSHRPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114380753-A Aryl or heteroaryl substituted quinoxaline-2, 3-diamine compound and antibacterial application thereof 中国医学科学院药物研究所 2022-04-22 CN claimed
CN-114380753-A Aryl or heteroaryl substituted quinoxaline-2, 3-diamine compound and antibacterial application thereof 中国医学科学院药物研究所 2022-04-22 CN disclosed