SCHEMBL29558696

SCHEMBL29558696

Fc1ccc(CNc2nc3ccccc3nc2NCc2ccc(F)cc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.63
KMT2A Q03164 3/20 0.63
MAPT P10636 2/20 0.63
LMNA P02545 1/20 0.63
APP P05067 1/20 0.63
KDM4E B2RXH2 2/20 0.58
NPSR1 Q6W5P4 1/20 0.58
HPGD P15428 1/20 0.58
PPARG P37231 1/20 0.58
NR2E3 Q9Y5X4 1/20 0.58
NCOR2 Q9Y618 1/20 0.58
TP53 P04637 1/20 0.54
POLB P06746 2/20 0.53
USP1 O94782 1/20 0.53
WDR48 Q8TAF3 1/20 0.53
KCNH3 Q9ULD8 3/20 0.53
MAPK1 P28482 1/20 0.50
USP10 Q14694 1/20 0.50
PIK3C3 Q8NEB9 1/20 0.50
USP13 Q92995 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29558388 0.89 APP (0.56) MEN1KMT2AMAPTLMNAAPP
SCHEMBL28725369 0.89 APP (0.56) MEN1KMT2AMAPTLMNAAPP
SCHEMBL29558267 0.84 LMNA (0.56) MEN1KMT2AMAPTLMNAAPP
SCHEMBL29558517 0.84 KDM4E (0.49) MEN1KMT2AMAPTLMNAAPP
SCHEMBL17432180 0.84 RAD52 (0.65) MEN1KMT2AMAPTLMNAAPP
SCHEMBL29558251 0.83 MAPT (0.49) MEN1KMT2AMAPTLMNAAPP
SCHEMBL29558864 0.81 APP (0.63) KMT2AAPPKDM4EPOLBUSP1
SCHEMBL19553913 0.80 APP (0.61) MEN1KMT2AMAPTLMNAAPP
SCHEMBL2590855 0.79 RAD52 (0.82) MEN1KMT2AMAPTLMNAAPP
SCHEMBL23657552 0.79 KDM4E (0.53) MEN1KMT2AMAPTLMNAAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114380753-A Aryl or heteroaryl substituted quinoxaline-2, 3-diamine compound and antibacterial application thereof 中国医学科学院药物研究所 2022-04-22 CN claimed
CN-114380753-A Aryl or heteroaryl substituted quinoxaline-2, 3-diamine compound and antibacterial application thereof 中国医学科学院药物研究所 2022-04-22 CN disclosed