SCHEMBL2955879

SCHEMBL2955879

Cc1ccc(-c2cccc(F)c2)c(C(=O)N2C[C@H]3C[C@H]3[C@H]2C(N)=O)c1

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 15/20 0.41
HCRTR1 O43613 14/20 0.41
CHRM3 P20309 3/20 0.38
GRM5 P41594 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2925061 0.92 HCRTR2 (0.41) HCRTR2HCRTR1CHRM3GRM5
SCHEMBL2929940 0.92 HCRTR1 (0.38) HCRTR2HCRTR1
SCHEMBL2928729 0.89 HCRTR1 (0.42) HCRTR2HCRTR1
SCHEMBL2929613 0.88 CHRM1 (0.44) HCRTR2HCRTR1
SCHEMBL3415999 0.88 HCRTR2 (0.48) HCRTR2HCRTR1CHRM3GRM5
SCHEMBL2931529 0.86 HCRTR1 (0.46) HCRTR2HCRTR1
SCHEMBL2927512 0.86 CYP46A1 (0.41) HCRTR2HCRTR1
SCHEMBL2926251 0.86 HCRTR2 (0.39) HCRTR2HCRTR1
SCHEMBL2955880 0.85 HCRTR2 (0.43) HCRTR2HCRTR1CHRM3
SCHEMBL2931039 0.85 HCRTR2 (0.39) HCRTR2HCRTR1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed