SCHEMBL29586646

SCHEMBL29586646

O=C(c1ccc(F)cc1)N1CCc2nc(-c3ccccn3)ncc2C1

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 2/20 0.68
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
TACR3 P29371 1/20 0.53
CYP2C19 P33261 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21326025 1.00 HSP90AB1 (0.68) HSP90AB1CYP1A2CYP2D6CYP2C9TACR3
SCHEMBL29587104 0.92 PDGFRB (0.58) HSP90AB1
SCHEMBL21326011 0.92 PDGFRB (0.58) HSP90AB1
SCHEMBL21325971 0.91 HSP90AB1 (0.56) HSP90AB1
SCHEMBL29586847 0.91 HSP90AB1 (0.56) HSP90AB1
SCHEMBL21325974 0.89 HSP90AB1 (0.68) HSP90AB1TACR3
SCHEMBL22295251 0.89 HSP90AB1 (0.54) HSP90AB1
SCHEMBL29587216 0.89 HSP90AB1 (0.68) HSP90AB1TACR3
SCHEMBL21326038 0.89 HSP90AB1 (0.54) HSP90AB1
SCHEMBL21326010 0.89 HSP90AB1 (0.54) HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110088103-B Novel tetrahydropyridopyrimidine compounds for the treatment and prophylaxis of hepatitis b virus infection 豪夫迈·罗氏有限公司 2022-04-12 CN claimed
CN-110088103-B Novel tetrahydropyridopyrimidine compounds for the treatment and prophylaxis of hepatitis b virus infection 豪夫迈·罗氏有限公司 2022-04-12 CN disclosed