SCHEMBL29600830

SCHEMBL29600830

C[C@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](C)NC(=O)[C@@H](N)CC(N)=O)C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 10/20 0.54
OPRM1 P35372 6/20 0.54
OPRK1 P41145 1/20 0.54
NPY4R P50391 2/20 0.50
NPY1R P25929 1/20 0.50
NPY2R P49146 1/20 0.50
CASP1 P29466 1/20 0.47
BACE1 P56817 2/20 0.47
MME P08473 1/20 0.46
ACE P12821 1/20 0.46
CPA1 P15085 1/20 0.46
ACE2 Q9BYF1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30420544 1.00 OPRD1 (0.54) OPRD1OPRM1OPRK1NPY4RNPY1R
SCHEMBL30086863 0.98 OPRD1 (0.53) OPRD1OPRM1OPRK1NPY4RNPY1R
SCHEMBL31614370 0.95 NPY4R (0.58) OPRD1OPRM1OPRK1NPY4RNPY1R
SCHEMBL30799508 0.92 OPRD1 (0.55) OPRD1OPRM1OPRK1NPY4RNPY1R
SCHEMBL30799878 0.91 OPRD1 (0.58) OPRD1OPRM1OPRK1BACE1MME
SCHEMBL29991172 0.90 OPRD1 (0.54) OPRD1OPRM1OPRK1NPY4RNPY1R
SCHEMBL29822851 0.88 OPRD1 (0.64) OPRD1OPRM1OPRK1NPY4RNPY1R
SCHEMBL30799540 0.88 OPRD1 (0.54) OPRD1OPRM1OPRK1CASP1BACE1
SCHEMBL29850189 0.87 OPRD1 (0.55) OPRD1OPRM1OPRK1NPY4RNPY1R
SCHEMBL31482982 0.87 NPY4R (0.57) OPRD1OPRM1OPRK1NPY4RNPY1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114605522-A MCL-1 and BCL-XL protein dual-targeting BH3 polypeptide mimics and application thereof 中山大学 2022-06-10 CN claimed
CN-114605522-A MCL-1 and BCL-XL protein dual-targeting BH3 polypeptide mimics and application thereof 中山大学 2022-06-10 CN disclosed