Methsergide

Methsergide

SCHEMBL29601488

CCC(CC)NC(=O)[C@@H]1C=C2c3cccc4c3c(cn4C)C[C@H]2N(C)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 10/20 0.91
ALDH1A1 P00352 9/20 0.91
MEN1 O00255 9/20 0.91
KDM4E B2RXH2 8/20 0.91
CYP2D6 P10635 7/20 0.91
HPGD P15428 7/20 0.91
HSD17B10 Q99714 7/20 0.91
MAPT P10636 5/20 0.91
HTR1A P08908 3/20 0.91
HTR2C P28335 3/20 0.91
HTR2B P41595 3/20 0.91
RECQL P46063 3/20 0.91
HIF1A Q16665 3/20 0.91
GLA P06280 2/20 0.91
ADRA2A P08913 2/20 0.91
DRD2 P14416 2/20 0.91
ADRA2B P18089 2/20 0.91
ADRA2C P18825 2/20 0.91
DRD1 P21728 2/20 0.91
HRH2 P25021 2/20 0.91

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methysergide SCHEMBL29359107 0.95 KMT2A (1.00) KMT2AALDH1A1MEN1KDM4ECYP2D6
Methysergide SCHEMBL467883 0.95 KMT2A (1.00) KMT2AALDH1A1MEN1KDM4ECYP2D6
Methysergide SCHEMBL41843 0.95 KMT2A (1.00) KMT2AALDH1A1MEN1KDM4ECYP2D6
Methysergide SCHEMBL467884 0.95 KMT2A (1.00) KMT2AALDH1A1MEN1KDM4ECYP2D6
Methysergide SCHEMBL28086572 0.94 KMT2A (0.98) KMT2AALDH1A1MEN1KDM4ECYP2D6
Methysergide SCHEMBL7088235 0.94 KMT2A (0.98) KMT2AALDH1A1MEN1KDM4ECYP2D6
Methysergide SCHEMBL41844 0.91 KMT2A (1.00) KMT2AALDH1A1MEN1KDM4ECYP2D6
Methysergide SCHEMBL29408580 0.91 KMT2A (1.00) KMT2AALDH1A1MEN1KDM4ECYP2D6
Methysergide SCHEMBL21803661 0.91 KMT2A (1.00) KMT2AALDH1A1MEN1KDM4ECYP2D6
Methysergide SCHEMBL28196309 0.91 KMT2A (1.00) KMT2AALDH1A1MEN1KDM4ECYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114146057-A Pharmaceutical composition and use thereof 斯皮内特赫拉公司 2022-03-08 CN disclosed