SCHEMBL29609013

SCHEMBL29609013

CNc1nc(N)nc(NCCc2ccccc2)n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 3/20 0.60
APP P05067 4/20 0.57
CA1 P00915 2/20 0.57
CA2 P00918 2/20 0.57
CA9 Q16790 2/20 0.57
BCHE P06276 2/20 0.57
ACHE P22303 2/20 0.57
CDK9 P50750 1/20 0.52
HDAC1 Q13547 1/20 0.52
ADORA2A P29274 3/20 0.51
ADORA2B P29275 3/20 0.51
ADORA1 P30542 3/20 0.51
ADORA3 P0DMS8 2/20 0.51
TMIGD3 P0DMS9 1/20 0.51
ADRA1D P25100 1/20 0.50
HTR2C P28335 1/20 0.50
ADRA1A P35348 1/20 0.50
ADRA1B P35368 1/20 0.50
HTR6 P50406 1/20 0.50
ACKR3 P25106 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14869438 1.00 HTR7 (0.60) HTR7APPCA1CA2CA9
SCHEMBL14869419 0.92 APP (0.65) HTR7APPCA1CA2CA9
SCHEMBL14869405 0.91 HTR7 (0.68) HTR7APPCA1CA2CA9
SCHEMBL2451092 0.89 APP (0.64) HTR7APPCA1CA2CA9
SCHEMBL14869457 0.86 APP (0.58) APPCA1CA2CA9BCHE
SCHEMBL14869402 0.85 NPSR1 (0.64) APPCA1CA2CA9BCHE
SCHEMBL29609599 0.85 NPSR1 (0.64) APPCA1CA2CA9BCHE
SCHEMBL1938196 0.84 HTR7 (0.56) HTR7APPCA1CA2CA9
SCHEMBL22151175 0.83 APP (0.64) APPBCHEACHEADORA2AADORA2B
SCHEMBL14869396 0.82 HPGD (0.62) HTR7APPCA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108191774-B Heterocyclic compound, preparation method and application thereof 中国药科大学 2022-05-24 CN disclosed